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N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4-trimethoxybenzamide
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-{5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
4-(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-1-yl)quinazoline
7-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidine
N-(2-chloro-4-fluoro-5-methylphenyl)-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-4-(pyridin-4-yl)piperazine-1-carboxamide
2-methyl-7-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-chloro-3-{[(1-methoxypropan-2-yl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
2-[4-cyclobutyl-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
N-{[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]methyl}acetamide
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
6-(4-cyanopiperidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-[(5-chlorofuran-2-yl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
(3S,5R)-1-(3-cyclopentylpropanoyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-methoxy-3-methyl-2-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}-1H-indole
3-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
(2R,3R)-N-(2-fluorophenyl)-2-hydroxy-3-[(2-hydroxyethyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-acetamido-N-(4-methoxyphenyl)-5-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]benzamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-fluoro-3-methoxybenzoyl)piperidine
N-(2H-1,3-benzodioxol-5-yl)-1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-3-amine
1-(4-methoxyphenyl)-4-[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]piperazine
3-(2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
N-[3-(azepan-1-yl)propyl]-N,1,5-trimethyl-1H-pyrrole-2-carboxamide
N,8-dimethyl-3-({[2-(2-oxopiperidin-1-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-(2-chlorophenyl)-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(2-cyclohexylethyl)-2-(pyridine-3-sulfonyl)-2,7-diazaspiro[4.5]decane
methyl 2-[methyl(2-phenylethyl)sulfamoyl]-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]-2-fluorophenol
N-(cyclopropylmethyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-(2-aminoethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-{2-methyl-6-[1-(pyrrolidin-3-ylmethyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
3-(thiomorpholine-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-one
4-chloro-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)benzamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
N-[1-(7-{[5-(hydroxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
[5-(1-benzofuran-5-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
4-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-(3-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]pyrimidine
(1s,4s)-4-hydroxy-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclohexane-1-carboxamide
(2S)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylamino)propan-1-one
(5S,9aS,9bS)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]acetamide
1-(propan-2-yl)-4-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-2-yl}piperidine