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(4aR,8aS)-6-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-benzyl-1-(quinolin-2-ylmethyl)piperidine-4-carboxylate
2-[2-(2-ethoxyphenyl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}quinoline
1-(carbamoylmethyl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]piperidine-3-carboxamide
3-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
6-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
2-[4-({4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
methyl 2-[4-(3,5-dimethyl-1H-indole-2-carbonyl)-2-oxopiperazin-1-yl]acetate
2-benzoyl-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
7-(propan-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}naphthalen-2-ol
(2S,4R)-1-cyclopentyl-N,N-diethyl-4-[5-(hydroxymethyl)furan-2-amido]pyrrolidine-2-carboxamide
N-(2-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(trifluoromethyl)pyrimidine
5-[1-(2-fluorobenzoyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
4-{1-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]propyl}pyridine
1-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
[(1-methyl-1H-pyrazol-4-yl)methyl]({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
1-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
1-[(4-fluorophenyl)methyl]-N-(1H-indol-2-ylmethyl)-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
1-(4-{[(3-methylpyrazin-2-yl)amino]methyl}phenyl)pyrrolidin-2-one
methyl 8-[(4-methoxy-2,3-dimethylphenyl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)thiomorpholine
3-cyclobutanecarbonyl-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(3R,4R)-1-{[5-(4-methylphenyl)furan-2-yl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(4-aminoazepan-1-yl)-2-(3,4,5-trimethoxyphenyl)ethan-1-one
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-2-(methylamino)pyridine-3-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[2-(difluoromethoxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-cyclopentanecarbonyl-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
8-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-{[(3-methoxyphenyl)formamido]methyl}-5-[2-(thiophen-3-yl)acetamido]benzoate
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]imidazolidine-2,4-dione
11-{[(2,3-difluorophenyl)methyl]amino}-4-[(2-methoxyphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-cyclopropyl-3-[5-(4-methyl-1H-imidazole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
[(2-chloro-6-fluorophenyl)methyl](ethyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-methoxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N3-ethylpiperidine-1,3-dicarboxamide
N-cyclopropyl-2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(1-benzothiophen-2-ylmethyl)(methyl){[4-({1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
5-amino-4-chloro-N-[3-(pyridin-3-yl)propyl]-1H-pyrazole-3-carboxamide
2-methyl-4-{4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
N-benzyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide