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7-(2-hydroxyethyl)-2-(3-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(4-methoxyphenyl)-4-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
2-{[5-(3-fluoropyridin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-(2-fluoroethyl)-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-ethanesulfonamido-N-(1-methoxypropan-2-yl)-1-methyl-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(3aR,6aR)-2-(oxan-4-yl)-5-(2,4,5-trifluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
methyl 8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrazine-2-carboxamide
ethyl 1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carboxylate
8-[3-(2-methylpropyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]quinoline
3-cyclopropyl-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
methyl({[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
[(2S,6S)-4-(3,4-dimethoxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
methyl 5-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[3-(cyclohexylsulfanyl)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[3-(pyridin-3-yloxy)propyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[(diethylcarbamoyl)methyl]-N-[(4-ethylphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-benzofuran-2-carboxamide
(2S)-3-hydroxy-2-[5-(5-hydroxy-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
N-ethyl-3-(2-methyl-1H-imidazol-1-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
methyl 3-cyclohexanecarbonyl-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-ethoxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
5,6-dimethyl-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-methyl-2-(morpholin-4-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
1-(4-fluorophenyl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclopropane-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
2-(dimethylamino)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
[(8-methoxy-2H-chromen-3-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-[(3,4-difluorophenyl)methyl]-4-(2,6-dimethylpyridin-4-yl)piperazine
2-cyano-N-[(2-ethoxyphenyl)methyl]-N-ethylbenzamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methyl-1,3-thiazole-5-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(piperidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-{4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]morpholin-3-yl}acetamide
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
methyl 3-(2,3-dimethoxybenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(3-phenylpropyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
N-(4-{4-[3-(morpholin-4-ylmethyl)phenoxy]piperidine-1-carbonyl}phenyl)acetamide
N2-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyrimidine-2,4-diamine
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
(2E)-3-(2,4-difluorophenyl)-1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)prop-2-en-1-one