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3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
N-cyclopentyl-3,4,5-trimethoxy-N-{[4-(oxolan-3-yloxy)phenyl]methyl}benzamide
1-methyl-4-{[5-(2-methylprop-1-en-1-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
1-methanesulfonyl-3-[2-(2-methylphenyl)ethyl]piperidine
N-[1-(4-chlorophenyl)ethyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
methyl(1,2-oxazol-5-ylmethyl){[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amine
N,N-dimethyl-2-(pyridin-3-yl)-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
(5S,9aS,9bS)-5-(1-ethyl-1H-pyrazol-4-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(1-methylpiperidin-4-yl)methyl]-2-oxo-N-(2-phenylethyl)-2-(pyridin-3-yl)acetamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-[4-(2-fluorophenyl)piperazin-1-yl]propan-1-one
4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-(thiophen-3-ylmethyl)piperidine
(1S,5R)-10-oxo-N-[3-(1,3-thiazol-4-yl)phenyl]-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
N-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
(isoquinolin-5-ylmethyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[4-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
2-{[benzyl(butyl)amino]methyl}-4-(pyrazin-2-yl)phenol
2-(2-fluorophenyl)-N-[2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-(2-phenylethyl)-1-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
4-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
{3-[5-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
2-(pyridin-3-ylmethyl)-4-(4-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
6-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-3-ol
N-[(7-{imidazo[1,2-a]pyridine-2-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
5-(2,6-dimethoxyphenyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-1H-imidazole
5-[3-(diphenylmethyl)-1,2-oxazole-5-carbonyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[2-(4-fluorophenyl)ethyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
11-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(1S,5R)-6-(2-methoxyethyl)-3-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-5-(2-methoxyacetamido)-N-methyl-N-[(4-methylphenyl)methyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]cyclobutanecarboxamide
5-(4-chloro-1-methyl-1H-pyrazol-5-yl)-3-methyl-1H-1,2,4-triazole
3-({3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1λ6-thiolane-1,1-dione
4-[5-(ethanesulfonyl)thiophen-2-yl]-1-methyl-1H-pyrazole
2-(cyclohex-1-ene-1-carbonyl)-1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-(azocan-1-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
dimethyl({2-[2-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]ethyl})amine
2-[4-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)-2-oxopiperazin-1-yl]benzonitrile
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(E)-2-phenylethenesulfonyl]piperidine
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
1-{2-hydroxy-3-[4-methoxy-2-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1-(azepan-1-yl)-3-{3-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenoxy}propan-2-ol
3-[2-(4-fluorophenyl)ethyl]-1-(5-methyl-1,2-oxazole-4-carbonyl)piperidine
3-cyclopropanecarbonyl-9-{[4-(prop-2-yn-1-yloxy)phenyl]methyl}-3,9-diazaspiro[5.5]undecane
4-[(2S)-2-amino-2-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)ethyl]phenol