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4-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-3,4-dihydro-2H-1,4-benzoxazine
(2E)-3-(3-fluorophenyl)-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}prop-2-enamide
2-{[(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
methyl 6-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4S)-4-amino-N-ethyl-1-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]pyrrolidine-2-carboxamide
1-{[({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)carbamoyl]methyl}piperidine-4-carboxamide
2-ethoxy-1-[1-(hydroxymethyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
methyl 4-{[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazol-7-yl]formamido}butanoate
1-[4-(aminomethyl)cyclohexanecarbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(4-fluorophenyl)methyl]-3-methyl-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
1-[(4aR,8aR)-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(4-methylphenoxy)ethan-1-one
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
(3aS,6aR)-5-(2-methylquinolin-4-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-cyclohexyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-hydroxy-2-(pyridin-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide
1-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-(3-methoxyphenyl)pyrrolidin-1-yl]acetamide
4-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
9-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]piperidin-4-amine
N-[1-({[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]propan-1-one
3-phenyl-N-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
(2S,4R)-N,N-diethyl-1-(1-methyl-1H-imidazole-5-carbonyl)-4-propanamidopyrrolidine-2-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
[1-(2,6-diaminopyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
2-[6-(methoxymethyl)pyrimidin-4-yl]-N,N-bis(propan-2-yl)benzamide
(1S,5R)-6-benzyl-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
3-[2-(3-fluorophenyl)acetyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-cyclopropyl-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[2-(2,3,6-trifluorophenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
5-cyano-N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(butan-2-yl)-N3-butyl-N5-(furan-2-ylmethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-({[(1S,2R)-2-(butylcarbamoyl)cyclohexyl]formamido}methyl)thiophene-2-carboxylic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
ethyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2-phenylpropyl)benzamide
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide