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N-cyclopropyl-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
[(4-methyl-1H-imidazol-5-yl)methyl](oxolan-2-ylmethyl)propylamine
N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N5-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-2-(2-methylfuran-3-amido)-7-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-(3-fluorophenyl)-1-methyl-3-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-methyl-9-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-{4-[(2-fluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(diphenylmethyl)-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-[4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1-(furan-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
N-(3-hydroxypropyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
6-[4-(hydroxymethyl)piperidin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
methyl (2S)-2-(3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-phenylpropanoate
1-(4-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}cyclopropane-1-carboxamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-1,3-thiazole-4-carboxamide
methyl 3-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-({7-[3-(furan-2-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
6-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
(3S,5R)-N-cyclohexyl-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
6-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
2-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
2-[benzyl(methyl)amino]-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-cycloheptyl-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
3-(1H-1,3-benzodiazol-1-yl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)propanamide
1-(6-methoxy-4-methylquinazolin-2-yl)-N-(2-methylpropyl)piperidin-4-amine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-3-yl)acetamide
N-[(3S,4R)-1-(cyclobutylmethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
ethyl 5-(2H-1,3-benzodioxol-5-yl)pyridine-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[3-(trifluoromethyl)phenyl]acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxyacetamide
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
[3-({[1-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-({[(3R,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(2R,3R)-1'-[(3-fluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
[(2-fluoro-5-methoxyphenyl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
ethyl 2-{1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}acetate
4-(1-butyl-1H-imidazol-2-yl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-ethyl-2-methylpyrimidin-4-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-methyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
N'-(2,5-dimethylphenyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanediamide