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methyl 1-({4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
6-ethyl-2-(morpholin-4-yl)-N-(pyridin-4-ylmethyl)pyrimidin-4-amine
2-(3-methoxyphenoxymethyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-{4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
2-methyl-3-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)quinoxaline
5-methyl-5-[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-4-yl]-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-[2-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(1S,5R)-6-[(3,4-difluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-chloro-4-hydroxyphenyl)-1-[3-(2-fluorophenyl)pyrrolidin-1-yl]ethan-1-one
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
3-{[(2-hydroxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(2,2-dimethyloxan-4-yl)-1-[4-(1H-imidazol-1-yl)phenyl]piperidin-4-amine
5-acetyl-N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
4-(benzyloxy)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2,4,5-trifluorobenzamide
3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(5-methylfuran-2-yl)benzamide
2-hydroxy-3,5-bis(propan-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
2-(4-methoxyphenyl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(thiophene-2-carbonyl)piperidine
N-[(5-ethylpyridin-2-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
9-(cyclopropylmethyl)-4-(ethanesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(4-hydroxypiperidin-1-yl)methyl]-6,8-dimethylquinolin-4-ol
(2R,6R)-4-(dimethyl-1,2-oxazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
6-(dimethylamino)-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
1-{3-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
2-(3,4-dimethoxyphenyl)-1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1H-imidazole
ethyl 1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-[(3R,4S)-1-{[(4-methylphenyl)methyl]carbamoyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1S,5R)-3-benzoyl-6-(2-ethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-(1,3-benzothiazol-2-yl)-4-[(2-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2,3-difluorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
3-(1H-indol-3-ylmethyl)-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(3S,4S)-4-methyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidine-3,4-diol
1-(2,2-dimethylpropanoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
4-[(2,6-difluorophenyl)methyl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-6,8-dimethyl-4-(thiophen-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
{3-[(3-chlorophenyl)methyl]-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}methanol
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[3-(ethoxymethyl)-4-methoxyphenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[4-(3-ethenylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-{[4-(2-methylphenyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-[(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]oxy}hex-5-en-1-yl)(methyl)amino]-N,N-dimethylacetamide
(2S,4R)-N,1-bis(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(4-chloro-3-methylbenzoyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-5-methoxy-1H-indole