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N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
5-[(3-methoxyphenyl)methyl]-3-methyl-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-(4-fluorophenoxy)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]acetamide
2-{2-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(1H-imidazol-2-ylmethyl)({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
2-amino-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-(oxolan-3-yl)pyridine-3-carbonitrile
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-N-(1,5-dimethyl-1H-pyrazol-4-yl)acetamide
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
2-{4-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
(1R,5R)-3-methanesulfonyl-N-(2-methoxy-5-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-benzyl-N-(cyclobutylmethyl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
(2R,6R)-10-methoxy-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{[1-(2,1-benzoxazole-3-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-6-methylpyrimidin-2-yl}phenol
3-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenol
2-[5-(2,2,3,3-tetramethylcyclopropanecarbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
(4-{[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methanol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
(3S,4S)-1-[6-(piperidin-1-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-(2-cyclopropylquinoline-4-carbonyl)-6-methyl-1-(2-methylphenyl)piperazin-2-one
2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
(2R,6S)-4-{3-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]-6-(2-methoxyphenyl)pyridin-2-yl}-2,6-dimethylmorpholine
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2-fluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(5S,9aS,9bS)-5-(3,5-dimethyl-1H-indol-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]methyl}-5,8-dimethyl-1,4-dihydroquinolin-4-one
(1S,5R)-3-benzoyl-N-(4-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
1'-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-benzyl-1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-[(2R,3R,6R)-5-(2-methoxypyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
6-methyl-2-(3-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-[4-({4-[5-(3-fluorophenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
3-{1-[2-(1,3-benzoxazol-2-yl)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(3-fluoro-4-methoxyphenyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1H-imidazol-1-ylmethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidine
N-(4-fluoro-2-methylphenyl)-2-({2-methylimidazo[1,2-a]pyrimidin-3-yl}formamido)propanamide
2-methyl-2-phenyl-N-[2-(pyridin-3-yloxy)propyl]propanamide
(1S,5R)-3-[(3-chloro-4,5-diethoxyphenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(azepan-1-yl)-2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
methyl 8-[(2,3-dimethoxyphenyl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
2-({6-[2-(trifluoromethoxy)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
N-[2-fluoro-5-(trifluoromethyl)phenyl]-2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carboxamide