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methyl (2S,4S)-1-(1-ethylpiperidin-4-yl)-4-(furan-2-amido)pyrrolidine-2-carboxylate
6-amino-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyridine-3-carboxamide
(1R,9aR)-1-{[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
6-butyl-2-[2-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
(5S)-5-[({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
1-cyclohexyl-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
8-(4-fluoro-2-hydroxyphenyl)-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
5-chloro-2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrrol-1-yl)pyridine
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
14-{2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-4-yl}-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{[2-(6-chloro-2-fluoro-3-methylphenyl)-1H-imidazol-1-yl]methyl}pyridine
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-phenylethyl)pyrimidine
N,4-dimethyl-4-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pentanamide
7-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
methyl 1-methyl-3-(3-phenylpropanamido)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
1-ethyl-3-(4-methylpiperazine-1-carbonyl)-N-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-ethylphenyl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
2-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}pyrimidine
2-(4-acetylphenoxy)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}cyclohexanecarboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-ol
8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
ethyl 1-(2-methoxyacetyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-[3-(3-fluorophenyl)phenyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
4-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(methylsulfanyl)pyrimidine
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
9-methoxy-4-(6-methoxypyrimidin-4-yl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[4-({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-1-yl]pyrazine-2-carbonitrile
N-({7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
methyl 5-{[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{3-[methyl(phenyl)amino]propyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
4-[3-(morpholin-4-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)quinoline
{1-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-(piperidin-1-yl)ethan-1-one
5-tert-butyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,3,4-oxadiazol-2-amine
4-methyl-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,3-thiazole-5-carboxamide
4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)benzoic acid
N-[(3-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 4-(4-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
2-({[(2-methylphenyl)methyl]sulfanyl}methyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-ethyl-6-methylphenyl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
2-cyclopropyl-N-[3-(methylsulfanyl)phenyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide