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N-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)-4-ethylcyclohexane-1-carboxamide
N-[5-(2-methanesulfonylacetamido)-2-methylphenyl]-4-methylbenzamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
5-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-[2-(2-chloro-4-fluorophenyl)acetyl]-1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-methoxyacetyl)-N-[2-(3-methylthiophen-2-yl)ethyl]piperidine-4-carboxamide
1-[4-({3-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
6-(1-cyclopentylpiperidine-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
4-(4-methylphenoxy)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine
2-oxo-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(3-methylbutyl)-8-(6-methylpyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2-fluorophenyl)-2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carboxamide
4-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-2-one
2-amino-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-methylpropanamide
4-benzoyl-1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
methyl 1-(benzyloxy)-2-oxo-8-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
4-hydroxy-N-(2-methoxybutyl)-2-(4-methylphenyl)pyrimidine-5-carboxamide
(4aS,8aR)-1-propyl-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-chloro-N-[(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]benzamide
1-[(2-fluorophenyl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-(2,3-difluorobenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[2-(piperidin-1-yl)ethyl]-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
5-methyl-2-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole
[(3-methyl-1,2-oxazol-5-yl)methyl](2-methylpropyl)(thiophen-3-ylmethyl)amine
6-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
(1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperidin-2-yl)methanol
1-{5-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
ethyl 1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxylate
2-({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(pyrrolidin-1-yl)butan-1-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-8-fluoroquinoline-2-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
N-[(2R,3R)-1'-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,4-dimethoxyphenyl)ethan-1-one
methyl (2S,4R)-4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-[(3-ethoxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
2-ethyl-9-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-[2-(3-phenylpiperidin-1-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
9-(5-methylpyridine-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-chlorophenyl)-4-[(5-fluoro-2-methoxyphenyl)methyl]-5-methylpiperazin-2-one
(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
(2R,6S)-4-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-2,6-dimethylmorpholine
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(2,5-dimethylphenyl)-3-({5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}formamido)propanamide
2-(3-chlorophenoxy)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
N-[2-(2-fluorophenyl)-1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-2-[(prop-2-en-1-yl)amino]benzamide
5-benzyl-5-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-4-(trifluoromethyl)benzamide