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4-{4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-(3-methoxyphenyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxamide
2-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methyl-1H-indole
[(3R,4S)-1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
9-(2-ethoxyethyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(3-methylphenyl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(5-methoxyfuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}quinoline
2-[2-(hydroxymethyl)phenyl]pyridine-4-carbonitrile
2-{3-[(3-chlorophenyl)methyl]-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})methylamine
methyl 1-(2-methoxyethyl)-5-[(6-methylhept-5-en-2-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(benzylsulfamoyl)[1-(thiophen-2-yl)propan-2-yl]amine
4-phenyl-3-(piperidin-3-yl)-1-(pyrimidin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-fluoro-5-methoxyphenyl)-1H-1,2,4-triazole-5-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}cyclopropanamine
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-yl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
(3R)-N-[(2-butoxy-3-methoxyphenyl)methyl]oxolan-3-amine
6-ethoxy-2-{4-[4-(4-methoxybenzoyl)piperazin-1-yl]piperidin-1-yl}-4-methylquinazoline
N-[(1-cyclobutylpiperidin-3-yl)methyl]quinoline-8-sulfonamide
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
4-({3-[3-(3,6-dimethylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-5-ethylfuran-2-carboxamide
4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
4-[1-(dimethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-1-(2-phenylethyl)piperidine
5-(2-phenylethyl)-5-[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-{imidazo[1,2-a]pyridin-2-yl}-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
N,N-dimethyl-4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-({3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(4-methylphenoxy)acetamide
N-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-1-cyclopentyl-6-oxopiperidine-3-carboxamide
1-[(2S)-2,3-dihydroxypropyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-4-[2-(1H-indazol-1-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethan-1-one
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(2-chloropyridin-3-yl)methyl]-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-cyclopropyl-4-[({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)methyl]pyrrolidin-2-one
N-[(3R,4S)-1-(3-hydroxypropyl)-4-phenylpyrrolidin-3-yl]-3-methanesulfonylpropanamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
N-[(4-phenyloxan-4-yl)methyl]-6-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
3-{1-[2-(4-fluorophenyl)ethyl]-1H-imidazol-2-yl}benzonitrile
ethyl 1-[(4-methoxyphenyl)methyl]-5-[3-(pyridin-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-benzyl-8-(cyclohex-3-en-1-ylmethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(piperazin-1-yl)ethyl]amino}methyl)piperidin-2-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(pyrrolidin-1-yl)pyridazine
ethyl 6-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-3-carboxylate