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2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-1-(pyridine-2-carbonyl)piperidine-4-carboxamide
(1r,4r)-4-[5-(2,1,3-benzoxadiazol-4-yl)-4-phenyl-1H-imidazol-1-yl]cyclohexan-1-ol
(2S,4S)-4-amino-N-ethyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidine-2-carboxamide
4-fluoro-N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}benzamide
5-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-methylpiperidine-2-carboxamide
[3-(cyclopropylmethyl)-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-3-yl]methanol
N,N-dimethyl-4-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}aniline
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-N-(4-fluorophenyl)piperidin-3-amine
3-(2-chlorophenyl)-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]propan-1-one
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
ethyl 4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-amido)piperidine-1-carboxylate
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propan-1-one
4-(1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)thiomorpholine
(1R,9aR)-1-({[3-(2-methoxyphenyl)propyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
3-(3-chlorobenzoyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(2R,3R)-1'-(2,5-dimethylfuran-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
4-({5-[1-(4-fluorophenyl)cyclopropyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
2-{5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-methyl-2-(4-methylpiperazin-1-yl)-N-(1,2-oxazol-3-ylmethyl)pyrimidine-5-carboxamide
7-(5-chloropyridin-2-yl)-4-[2-(1-methylpyrrolidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-chlorophenyl)-4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-2-one
4-benzyl-1-methyl-3-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-methyl-4-{4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]phenyl}butan-2-ol
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
1-[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
5-methoxy-N,3-dimethyl-N-(pyrazin-2-ylmethyl)-1H-indole-2-carboxamide
N-benzyl-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-N-methylpiperidin-3-amine
4-[4-(azepane-1-carbonyl)piperidin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(2-chlorophenyl)-4-{1-[4-(piperidin-1-ylmethyl)benzoyl]piperidin-3-yl}pyrimidine
2-[(4aR,7aS)-6,6-dioxo-4-(pyrrolidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
6-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[2-(2,3-dimethylphenoxy)acetyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({[cyclopropyl(3-methylpyridin-2-yl)methyl]carbamoyl}amino)-N-(2-methylpropyl)benzamide
8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{4-benzyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methanol
2,6-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyridine-4-carboxamide
4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(2-methoxyphenyl)piperazin-2-one
6-(aminomethyl)-N-[2-(4-fluorophenyl)ethyl]-2-methylpyrimidin-4-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(3-hydroxypiperidin-1-yl)ethan-1-one
1-[4-(1-methyl-4-phenyl-1H-imidazol-5-yl)phenyl]-1H-1,2,4-triazole
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol