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5-(2-chlorophenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]furan-2-carboxamide
3-{4-[(3-hydroxyphenyl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
ethyl 3-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]amino}propanoate
(1,4-dioxan-2-ylmethyl)(methyl)({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
methyl 2-chloro-4-({methyl[1-(methylcarbamoyl)propan-2-yl]carbamoyl}amino)benzoate
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
3,5-difluoro-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
2-[2-(4-propylpiperazin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
6-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-N-methylpyridine-2-carboxamide
methyl (2S)-2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanoate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,8-naphthyridine-2-carbonyl)piperidin-3-ol
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[(2-{4-[1-(piperidin-1-yl)ethyl]phenyl}phenyl)methyl]propanamide
3-(3-methoxyphenyl)-5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-[3-(methanesulfonylmethyl)piperidine-1-carbonyl]phenol
N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(2S)-1-acetyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrrolidine-2-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(5-chlorothiophen-2-yl)methyl]acetamide
2-cyclopropyl-9-(1H-imidazol-2-ylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,4S)-5-(2-acetylbenzoyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]piperazine
3-(1H-1,2,3-benzotriazol-4-yl)-1-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)urea
8-methoxy-5-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}quinoline
9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-6-(methoxymethyl)pyrimidin-4-amine
{[5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)thiophen-3-yl]methyl}dimethylamine
N-methyl-N-(1-methylpiperidin-4-yl)-3-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}propanamide
3-(diethylamino)-1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)propan-1-one
8-(1-methylcyclopropanecarbonyl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}isoquinoline
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)quinoline-2-carboxamide
4-fluoro-3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]benzene-1-sulfonamide
5-{1-[2-(4-chloro-2-methylphenoxy)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl){[2-(methylsulfanyl)phenyl]methyl}amine
5-methoxy-N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]furan-2-carboxamide
3-[1-(8-fluoroquinoline-2-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
1-tert-butyl-3-cyclopentyl-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
6-(4-methanesulfonylpiperazin-1-yl)-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-amine
3-methoxy-1-(4-{4-[(3R)-3-methylpiperazine-1-carbonyl]phenoxy}piperidin-1-yl)propan-1-one
2-{[cyclohexyl(thiophen-2-yl)methyl]amino}propane-1,3-diol
6-[3-(dimethylamino)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)-4-(pyrrolidine-1-carbonyl)pyrrolidine-2-carboxylic acid
2-(3-fluorophenoxymethyl)-8-(pyridazine-4-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-cyclohexyl-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}furan-2-carboxamide