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4-(4-fluoro-2-{[2-(thiophen-3-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzamide
3-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}propan-1-ol
4-fluoro-N-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
2,6-dimethyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]quinoline
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-[2-(difluoromethoxy)benzoyl]-4-[(4-fluorophenyl)methyl]-1,4-diazepane
methyl 6-[2-({2-[4-(methylsulfanyl)phenyl]acetamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxylate
methyl 2-({3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)acetate
1-(2-ethoxyethyl)-5-[4-(2-hydroxypropan-2-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(1H-pyrazol-1-yl)-1-[4-(thiophen-2-yl)butanoyl]piperidine-4-carboxylic acid
3-(2,5-difluorobenzoyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6-(1-cyclopentyl-5-oxopyrrolidine-3-carbonyl)-N,N,1-trimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-[(3S,4R)-3-(5-methylfuran-2-yl)-4-(oxane-4-amido)pyrrolidin-1-yl]propanoic acid
6-methoxy-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
2-(4-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-1,4-diazepan-1-yl)-1,3-benzoxazole
(2E)-3-(4-methoxyphenyl)-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{[1-(cyclopropylmethyl)piperidin-4-yl]methyl}acetamide
2-(3-chlorophenyl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
5-fluoro-2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
6-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1,4-oxazepan-6-ol
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
2-[(1S,5R)-6-[2-(2-fluorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
7-acetamido-N-(2-hydroxyethyl)-N-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
ethyl 4-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-3-yl]piperazine-1-carboxylate
4-benzyl-1-[(3-methoxyphenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-chloro-4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]cyclobutanecarboxamide
3-(2-ethylbutanoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(4-methoxyphenyl)methyl]-4-(oxolane-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(2-hydroxyphenoxy)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
(2E)-3-(2,3-difluorophenyl)-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
(5S)-5-{4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-methyl-2-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
dimethyl[(5-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]amine
methyl N-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}carbamate
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-methanesulfonylpropanamide
3-[4-(3-methylphenyl)piperazin-1-yl]-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}propan-1-one
2,6-difluoro-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-3-yl)propanamide
3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(thiophen-2-yl)ethyl]propanamide