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2-[1-(2,2-dimethylpropyl)-4-[(8-fluoroquinolin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
3-({[1-(furan-2-yl)ethyl]amino}methyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-benzyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-benzoxazole-5-carboxamide
[(3S,5R)-1-(5-chloropyridin-2-yl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
2-chloro-N-(2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)benzamide
(1S,5R)-3-[(2,4-dimethoxy-3-methylphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
9-[2-(2-methylpiperidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-methoxypiperidin-1-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
8-methoxy-2-[4-(2-methylphenoxy)piperidin-1-yl]quinoline
2-(4-methoxyphenyl)-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
3-{[(1R,3S)-3-(ethylcarbamoyl)-1,2,2-trimethylcyclopentyl]formamido}propanoic acid
2-{5-cyclopropyl-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-methoxyphenyl)pyrimidine
4-methoxy-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-benzyl-8-[(3,4-dimethoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
methyl 2-{[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}acetate
1-[2-(adamantan-1-yl)propan-2-yl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-[(1-ethylpiperidin-3-yl)methyl]-3-(4-methoxy-2-methylphenyl)urea
5-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)pyrimidin-2-amine
3-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)pyridin-2-ol
6-[(5-chloro-2-hydroxyphenyl)methyl]-N-(3,5-dimethylphenyl)-6-azaspiro[2.5]octane-1-carboxamide
2-ethoxy-N-[(1-methylpiperidin-3-yl)methyl]acetamide
3-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}benzoic acid
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
1-{3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}-1H-1,2,3,4-tetrazole
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-benzyl-1H-pyrazol-5-yl)acetamide
4-[2-(3,5-difluorophenyl)acetyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-(1H-pyrazol-1-yl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-methyl-6-[4-(oxan-4-yl)piperazin-1-yl]-2-phenylpyrimidine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[4-(3-fluorophenyl)phenyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
4-(azocan-1-yl)-N-(furan-2-ylmethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
5-chloro-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-3-carboxylic acid
(2E)-N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
4-chloro-1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-(3-chloro-4-methoxyphenyl)propanamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
4-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-methoxypyridine-3-carbonitrile
1-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]cyclopropane-1-carboxamide
1-{2-[5-(azocane-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}-2-ethoxyethan-1-one
5-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-2,1,3-benzoxadiazole
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-2,3-dihydro-1H-indazol-3-one
ethyl 2-(1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazol-6-yl}-N-methylformamido)acetate
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide