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({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
1-methyl-4-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-hydroxy-2-methylpropanoyl)piperidine-4-carboxamide
N-[(2R,3R)-1'-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
methyl 4-[6-(benzyloxy)-3-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]benzoate
(3-ethyl-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidin-3-yl)methanol
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
3-methoxy-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
N-(2-methyl-1-{7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
1-benzyl-3-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-[(3-ethoxy-4-methoxyphenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-hydroxy-5-methoxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
ethyl 1-(oxane-4-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
(3aR,7aS)-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]propanamide
2-cyclopentyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-1'-(thiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylpyrimidine
(3R,5S)-N-[3-(1H-imidazol-1-yl)propyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
1-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}pyrrolidin-3-yl)piperidine
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(9aS)-2-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
1-(3-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
2-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
7-acetamido-N-[(4-fluorophenyl)methyl]-N-methyl-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxamide
(2E)-3-(3,4-difluorophenyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}prop-2-en-1-one
(3E)-N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N-methylpent-3-enamide
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-[(3-hydroxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(morpholin-4-yl)benzamide
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]acetamide
2-(4-methoxyphenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-3,4-dimethoxybenzamide
N-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione