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3-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
2-(2-chlorophenyl)-N-(2-ethoxyethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenyl]imidazolidine-2,4-dione
N-cyclopentyl-4-methoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(2-oxo-2H-chromene-3-carbonyl)piperidine-3-carboxylate
1-cycloheptyl-N-methyl-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(2-chlorophenyl)methyl]-4-{3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-chloro-N-(oxolan-2-ylmethyl)-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
3-[(4-ethoxyphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
5-(2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-3-phenyl-1,2,4-oxadiazole
4-(3-{[1-(piperidin-3-yl)piperidin-4-yl]oxy}benzoyl)morpholine
3-methyl-1-[1-(6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
2-methoxy-1-{4-[(5-phenylthiophen-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-phenyl-4-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidine-1-carboxamide
1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
N-[2-(1H-indol-3-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-[2-(2-ethylpyrimidin-5-yl)-7,8-dimethylquinoline-4-carbonyl]piperidine-4-carbonitrile
1-{1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}-2-(3-methylphenyl)ethan-1-one
3-cyclohexyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
3-[(1H-imidazol-2-ylmethyl)(methyl)sulfamoyl]-N-phenylbenzamide
(3R,9aR)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-7-methylquinolin-3-yl}methanol
7-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(2-oxoazepan-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-(butan-2-yl)-2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
3-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-1-(morpholin-4-yl)propan-1-one
9-(2,1,3-benzoxadiazole-4-sulfonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(4aS,7aR)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
7-(2-hydroxyethyl)-2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
3-{2-oxo-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methyl-1,2-dihydrophthalazin-1-one
N-cyclobutyl-2-(oxane-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[2-(dimethylamino)ethyl]-6-oxo-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
5-methoxy-2-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}pyridin-4-ol
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclopropane-1-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-3-carboxylate
N-cyclopropyl-3-{1-[2-(4-phenylpiperidin-1-yl)acetyl]piperidin-4-yl}propanamide
N-(1-hydroxybutan-2-yl)-5-methyl-2-phenyl-N-(pyridin-3-ylmethyl)-1H-imidazole-4-carboxamide
1-(benzyloxy)-8-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1,8-diazaspiro[4.5]decan-2-one
N-benzyl-1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methylpiperidine-3-carboxamide
4-chloro-5-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine