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N-({7-[2-(3-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
2-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
6-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]propanamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(2,4-difluorophenyl)methyl]-1H-pyrazole-4-carboxamide
N,N-dimethyl-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
4-methyl-6-(4-{[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
3-(2-aminoethyl)-4-cyclohexyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[3-(dimethylamino)pyrrolidin-1-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
6-fluoro-2-[({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)methyl]quinolin-4-ol
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
(3S,9aR)-8-(3,5-difluorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-(naphthalen-1-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
1-[2-methoxy-5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
4,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-2-amine
N5-(3-methoxypropyl)-N6-(1-propylpiperidin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(2E)-3-(furan-2-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]prop-2-en-1-one
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[(5-methylthiophen-2-yl)methyl]amine
2-{5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-6-methylpyridine
3-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{9-[(4-fluoro-3-methoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
4-methoxy-N-(2-methoxyethyl)-2-{[1-(naphthalen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
(3S,4R)-4-(2-methylphenyl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
7-(2,3-dimethylbenzoyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1'-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
1-(2-methoxybenzoyl)-4-{3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}piperazine
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyridin-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-6-({3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)pyridine
1-[(3-fluorophenyl)methyl]-6-oxo-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
2-({[(3R,4R)-1-[(3-chloro-2,4-difluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
ethyl 4-{3-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]benzoyl}piperazine-1-carboxylate
methyl 3-cyclopropanecarbonyl-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{4-cyclopentyl-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-methylthiophene-2-carboxamide
3-[(4-methoxyphenyl)methyl]-8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-4-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}propan-1-one
4-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazine-1-carbaldehyde
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2R,6S)-4-{1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2,6-dimethylmorpholine
1-[(5-ethylpyridin-2-yl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[2-amino-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-phenylpiperidin-4-yl]ethan-1-one