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methyl 5-[(1-hydroxypropan-2-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
4-ethyl-3-(piperidin-4-ylmethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[cyclopropyl(ethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(6-methoxy-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)pyrrolidine-2-carboxamide
2-[2-methyl-3-({[1-(3-phenylpropyl)piperidin-3-yl]amino}methyl)-1H-indol-1-yl]acetamide
N-{[1-(morpholine-4-carbonyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-[1-(3-methylphenyl)piperidin-4-yl]acetamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
3-{2-[4-cyclohexyl-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
(3-{2-[1-(3-methoxypyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrazin-2-ol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(2-methoxyphenyl)-1H-pyrazole
5-(3-methoxy-2-methylphenoxymethyl)-3-(thiophen-2-yl)-1,2,4-oxadiazole
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-(3-methoxypropyl)-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3,5-dimethyl-1-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl)-1H-pyrazole
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-4-methyl-1,3-oxazole-5-carboxamide
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
4-phenyl-3-(piperidin-4-yl)-1-[3-(pyridin-3-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(4-{spiro[indene-1,4'-piperidine]-1'-yl}piperidin-1-yl)phenyl]pyridine-4-carboxamide
1-{1,3-dioxo-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(2-hydroxy-2-phenylethyl)-N-methylpiperidine-4-carboxamide
3-methyl-3-phenyl-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidine
4-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-imidazole
methyl 3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidine-1-carboxylate
2-(3-methoxypropyl)-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-(1-methyl-1H-imidazol-2-yl)-6-[4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
4-[1-(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
2-chloro-N-({1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}methyl)benzamide
4-{2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carbonyl}piperazin-2-one
2-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
ethyl 4-{6-[(3-ethoxy-4-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-cyclopropyl-4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
1-(4-phenylpiperazine-1-carbonyl)-6-{[4-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane
1-cyclohexyl-4-(3-phenyl-1,2-oxazole-5-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-2-(dimethylamino)acetamide
5-oxo-N-[3-(pyridin-2-yl)propyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-(4-{4-[(butan-2-yl)amino]piperidin-1-yl}phenyl)-4-methoxybenzamide
3,5-dimethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1-benzofuran-2-carboxamide
({4-ethyl-5-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(butan-2-yl)-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)-N-(pyridin-4-ylmethyl)acetamide
2-(3,4-dimethoxyphenyl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
2-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidine-1-carbonyl]-4H-chromen-4-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(quinolin-8-yl)urea
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane