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(1R,5R)-6-(cyclobutylmethyl)-3-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-({2-methoxy-5-[(3-phenoxyazetidin-1-yl)methyl]phenyl}methyl)pyrrolidine
3-(4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1H-pyrazole
8-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidine-4-carbonyl)morpholine
7-(2-methoxyacetamido)-1-methyl-N-[(1R,2S)-2-phenylcyclohexyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazole-5-carboxamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})amine
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(3R,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
4-(3-ethoxy-4-methoxyphenyl)-5-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2R)-2-amino-4-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pentanamide
2-(3-fluoro-4-hydroxyphenyl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
methyl 8-(1H-indol-3-ylmethyl)-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
4-{4-[(2-chlorophenyl)methyl]-4-(ethoxycarbonyl)piperidine-1-carbonyl}pyridin-1-ium-1-olate
4-(2-fluorophenoxy)-1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
2-methyl-4-[1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]cyclopent-1-ene-1-carboxamide
3-(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)prop-2-yn-1-ol
7-[(2-fluorophenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-[4-(6-cyclopropylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]propane-1,3-diol
2-amino-4-(isoquinolin-5-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
N'-(3-fluorophenyl)-N-[(1-propylpiperidin-3-yl)methyl]ethanediamide
2-[1-(2-methylphenyl)-5-[2-(1-methylpiperidin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[2-(pyridin-2-yl)ethyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-chlorophenyl)-4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
(3R,4R)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3,4-dimethylpyrrolidin-3-ol
4-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
7-(2-methoxyethyl)-N-(2-methoxyphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
9-(4,6-dimethylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
7-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-[2-(3-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]morpholine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-methyl-N-(thiophen-3-ylmethyl)propanamide
methyl 9-[3-(dimethylamino)propoxy]-3-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,5R)-N3-cyclopropyl-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
2-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-6,7-dimethoxyquinazolin-4-amine
3-(5-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
4-[5-(morpholine-4-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
4-[(2-fluorophenyl)methyl]-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,4-diazepan-5-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
[3-({1-[6-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-cyclohexyl-N-methyl-1,3-benzoxazole-6-carboxamide
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)piperidine
1-{2-[({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)amino]ethyl}pyrrolidin-2-one
N-[(2,5-difluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
(2S)-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-methyl-2-phenylpiperazine
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(1H-pyrazol-4-yl)butanamide