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N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amine
1-[(4-methylphenyl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-one
3-acetamido-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}propanamide
2-(1-{[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
2-{2-[3-(2-fluorophenoxy)azetidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N-(pyridin-3-yl)propanamide
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyridine-4-carboxamide
(1S,5R)-6-benzyl-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
9-methoxy-3-(6-methylpyridine-3-carbonyl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-({8-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
N-[(5-methylfuran-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(pyridin-3-yl)acetamide
1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-ethylpiperidine-4-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-{[(5-methylpyrazin-2-yl)methyl]amino}pyridine-3-carboxamide
4-benzyl-3-ethyl-1-(4-fluoro-3-methoxybenzoyl)-1,4-diazepan-5-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
N-[4-(3-fluorophenyl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxamide
N-[2-(2-chlorophenyl)ethyl]-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
4-{1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}benzoic acid
1-methyl-9-(prop-2-en-1-yl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylisoquinoline-5-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-diphenylacetamide
4-acetyl-N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)benzamide
{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methanamine
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N-(1-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
4,4,4-trifluoro-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
3-(4-hydroxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
1-(2,6-difluorobenzenesulfonyl)-2-(furan-2-yl)azepane
N-(1-methoxypropan-2-yl)-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N,N-dimethyl-2-[(1S,5R)-6-[(2E)-3-phenylprop-2-enoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-(1H-imidazol-1-ylmethyl)-1-(3,3,3-trifluoropropyl)piperidine
1-[(4-chlorophenyl)methyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
(2S,4R)-4-amino-1-(1-benzoxepine-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
[(3R,4R)-1-(2-fluoro-6-methoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[2-(2,4-difluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
1-(3-chlorophenyl)-4-({3-[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-2-yl)ethoxy]phenyl}methyl)piperazine
3-(4-methoxyphenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
4-(2-aminoacetyl)-5-benzyl-1-(4-methylphenyl)piperazin-2-one
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
2-[1-(hydroxymethyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
9-[2-(2-chlorophenoxy)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
3-(2,5-dioxoimidazolidin-4-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]propanamide
6-methyl-2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole