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3-chloro-2-fluoro-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
(4S,6R)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
5-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
2-[(3-methoxyphenyl)methyl]-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]azepan-3-amine
1-tert-butyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
ethyl 1-(2-phenylethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(dicyclopropylmethyl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperazine-1-sulfonamide
{4-[(8-methoxy-2H-chromen-3-yl)methyl]-1,4-oxazepan-6-yl}methanol
N-(2-hydroxyethyl)-4-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyridine-2-carboxamide
2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-phenyl-1,2,3,6-tetrahydropyridine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(4-methoxyphenyl)acetamide
3-(2-chlorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-chloro-N-cyclopentyl-4-({1-[(3-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
6-fluoro-8-[4-(piperidine-1-carbonyl)pyridin-2-yl]quinoline
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
N-[(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(thiophen-3-yl)acetamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-(propan-2-yl)-1,2-oxazole
N-[(2R,3R)-2-methoxy-1'-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
9-methoxy-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3-chlorophenyl)methyl]-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(methylsulfanyl)pyridine-3-carboxamide
2-(3-phenylpropyl)-4-(4,4,4-trifluorobutyl)morpholine
methyl 4-{[(2-{5-oxo-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
ethyl 4-(cyclopropylmethyl)-1-(naphthalene-1-carbonyl)piperidine-4-carboxylate
5-ethyl-2-methyl-4-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
5-(2-methylpropyl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-3-carboxamide
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrrolidine-2,5-dione
1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2,2-dimethyloxan-4-yl)-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(2,4-dihydroxyphenyl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
6-[2-(2,5-dimethoxyphenyl)acetyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(2,2-dimethylpropanoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
2-(2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-{5H,6H-imidazo[2,1-b][1,3]thiazole-3-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(furan-2-yl)ethyl]piperidine-3-carboxamide
1-(1-benzothiophen-2-ylmethyl)-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][(3-methyl-1-benzofuran-2-yl)methyl]amine