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1-(butane-1-sulfonyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
N-(4-{4-[(3,3-dimethylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
1-(2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}ethyl)piperidin-2-one
3,5-dimethyl-7-(5-methyl-2-phenylfuran-3-carbonyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
methyl 6-[(4-acetylpiperazin-1-yl)methyl]-3-(2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-methyl-3-(1-phenyl-1H-pyrazol-5-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
N-(oxan-4-yl)-3-[(pyridin-3-ylmethyl)sulfamoyl]benzamide
N,N-dimethyl-2-[4-(morpholine-4-carbonyl)pyridin-2-yl]aniline
(2E)-3-(3,4-difluorophenyl)-N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)prop-2-enamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(3,5-dimethoxyphenyl)methyl]piperidine
8-chloro-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]quinoline-2-carboxamide
2-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-(2-aminoethyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
ethyl 1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N,N-dimethyl-2-{[(3-methylphenyl)methyl]amino}-1-propyl-1H-1,3-benzodiazole-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
methyl 2-(4-benzyl-3-methyl-2-oxopiperazin-1-yl)acetate
3-(3-ethylphenoxy)-1-(7-methyl-1-benzofuran-2-carbonyl)azetidine
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-[2-oxo-2-(3-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopentanecarbonyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
1-[(4-fluoro-2-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-(2-hydroxyphenoxy)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
4-chloro-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrrole-2-carboxamide
N-methyl-2-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
(2S,4R)-4-amino-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-4-[1-(5-methylpyridine-3-carbonyl)piperidin-3-yl]-6-(pyrrolidin-1-yl)pyrimidine
7-(4-chloro-1H-pyrazole-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-(benzyloxy)-4-(2-chloro-6-fluorobenzoyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]propanamide
2-[4-(cyclohexylmethyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-methyl-N-(piperidin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
2-methyl-4-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-dihydrophthalazin-1-one
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3S)-2-oxoazepan-3-yl]propanamide
4,5-dimethyl-6-{4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}pyrimidine
({4-[1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methylpiperidin-4-amine
N-[4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
4-ethyl-3-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(isoquinoline-3-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
N-[2-(diethylamino)ethyl]-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-{ethyl[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]amino}-1λ6-thiolane-1,1-dione
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl}){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine