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N-(2-cyclohexaneamido-5-methylphenyl)oxolane-3-carboxamide
2-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-[2-(3-fluorophenyl)ethyl]-N-[2-(1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
methyl 5-{[(2-chlorophenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(diphenylmethyl)({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 6-{[(1-hydroxybutan-2-yl)(pyridin-3-ylmethyl)amino]methyl}pyridine-2-carboxylate
5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
4-methyl-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1H-imidazole-5-carboxamide
3,3-dimethyl-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]pyrrolidin-2-one
2-phenyl-7-(3-propyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-methoxy-4-oxo-N-[1-(phenylcarbamoyl)piperidin-4-yl]-1,4-dihydropyridine-2-carboxamide
5-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
(1,3-benzothiazol-2-ylmethyl)(methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][4-methyl-4-(methylsulfanyl)pentan-2-yl]amine
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4-chloro-2,5-dimethoxyphenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
1-[2-(2-chloro-4-fluorophenyl)acetyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl][(2-{[3-(trifluoromethyl)phenyl]methoxy}-6H,7H,8H-cyclopenta[g]quinolin-3-yl)methyl]amine
ethyl 1-ethyl-5-[3-(4-fluorophenyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(4-methanesulfonylphenyl)-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-cyclohexyl-4-[2-(1H-imidazol-2-yl)benzoyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
3-chloro-N-cyclopentyl-4-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-(4-fluorobenzoyl)-6-azaspiro[2.5]octane
2-(dimethylamino)-2-(2-fluorophenyl)-1-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}ethan-1-one
1-methyl-2-oxo-8-(1H-pyrazole-4-sulfonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(dimethylamino)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
3-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)benzonitrile
4-(3-hydroxy-3-methylbutyl)-N-[2-(pyrrolidin-1-yl)propyl]benzamide
8-(cyclohex-3-en-1-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(4-chloro-2-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
7-(5-chloropyridin-2-yl)-4-(5-fluoropyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[1-(3-chlorophenyl)-5-(oxolan-3-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
2-ethyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-(thiophen-3-ylmethyl)urea
7-methoxy-3-[(4-methoxypiperidin-1-yl)methyl]-2-(3-methylphenyl)quinoline
1-(cyclohex-1-ene-1-carbonyl)-3-(3,4-dimethoxybenzoyl)piperidine
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
7-(cyclobutylmethyl)-2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
N-[2-(4-sulfamoylphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-(1-methyl-1H-pyrazol-5-yl)-2-[4-(quinolin-2-yl)-1H-pyrazol-1-yl]acetamide
N-{[3-methyl-7-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
methyl 1-[(3R,5S)-1-[(2-fluorophenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-benzyl-4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one