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{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(2-methylpropyl)(pyridin-2-ylmethyl)amine
(3R,4R)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
ethyl 1-[3-(methylsulfanyl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
N-cycloheptyl-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}acetamide
1-[4-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
7-chloro-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-3-methyl-1H-indole
4-benzyl-3-ethyl-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
5-acetyl-6-methyl-3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1'-(2,1,3-benzoxadiazol-4-ylmethyl)-5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
N-{1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]piperidin-4-yl}methanesulfonamide
2-(2-methoxyethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-methoxyphenyl)methyl]-4-{1-oxa-7-azaspiro[3.5]nonan-7-yl}pyridine-2-carboxamide
N-methyl-1-(piperidin-3-ylmethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(4-methylpiperazin-1-yl)-3-{4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
N-(1-{1-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
5-{[3-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(1S,5R)-3-[(3-chlorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-fluorophenyl)-4-({4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
methyl 3-[4-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-1H-pyrazol-1-yl]propanoate
2-{4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
6-chloro-2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3,3-dimethyl-1-({5-[(3,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
2-[3-({[4-(furan-2-yl)butan-2-yl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
4-(2-fluorophenoxy)-1-[3-(1-methylcyclopropyl)propanoyl]piperidine-4-carboxylic acid
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxy-3-methoxypropyl)-5-methoxybenzamide
N-(1H-indol-3-yl)-1H-pyrazole-4-carboxamide
4-[(2R,3R)-1'-(2-cyclopentylacetyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-ol
(2R)-2-amino-N-(3-methoxy-2,2-dimethylpropyl)-2-phenylacetamide
4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-amino-6-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(dimethylamino)pyridine-3-carboxamide
N-{[7-(3-methylthiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}cyclopropanecarboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S)-2-amino-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-4-yl)-N-methylpropanamide
4-{[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
N-[(3-chlorophenyl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
3-(3-methyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}propanamide
N-[3-(2,6-dimethylphenoxy)propyl]-N,2-dimethylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-6-oxa-9-azaspiro[4.5]decane
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}pyrimidine
4-[2-(methylsulfanyl)propyl]-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-1,2,3-triazole
2-(3-fluorophenoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide