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N-[2-methoxy-5-({[(5-methyl-1H-imidazol-4-yl)methyl]carbamoyl}amino)phenyl]propanamide
5-(1-benzofuran-2-yl)-N-[2-(diethylamino)ethyl]-1,2,4-triazin-3-amine
N-(3-chloro-4-methoxyphenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
2-(2-chloro-6-fluorophenyl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-cyclopropyl-3-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
1-(4-fluorophenyl)-4-[3-(1H-imidazol-2-yl)piperidin-1-yl]butane-1,4-dione
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
5-[(dimethylsulfamoyl)amino]-1-methyl-N-(2-methylbutyl)-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
2-{4-[(2,6-dimethoxyphenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
2-{4-[4-(3-benzoylpiperidin-1-yl)piperidin-1-yl]phenyl}-N-(pyridin-2-ylmethyl)acetamide
1-[3-cyclopentyl-5-(5-methoxy-1H-indol-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
(1S,4R)-4,7,7-trimethyl-1-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-oxabicyclo[2.2.1]heptan-3-one
(3R,4R)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
methyl 3-acetamido-5-[(naphthalen-1-ylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4R)-4-amino-N-ethyl-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[2-(thiophen-2-yl)azetidin-1-yl]propan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-methyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-pyrazole
methyl 1-[(3S,5S)-1-(2-ethylbutyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-N-[2-(methylsulfanyl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2-phenylpropyl)-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
(4-{[1-(3-fluoropyridin-4-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-{[4-(propan-2-yl)phenyl]methyl}-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
4-(2-methyloxolane-2-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1R,3S)-7-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-7-azaspiro[3.5]nonane-1,3-diol
N-[2-(1-methyl-1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
3-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N,N-diethyl-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-tert-butyl-4-hydroxy-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
(3S,4S)-1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[4-(furan-3-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-3-methylbenzamide
3-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridin-2-amine
3-(2-fluorophenyl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-1-(4-methylphenyl)piperazin-2-one
7-acetamido-1-[2-(pyridin-2-yl)ethyl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
1-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
9-methoxy-3-[(5-methylthiophen-2-yl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(1H-1,3-benzodiazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[4-chloro-2-({4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetic acid
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-2-(3-methoxyphenyl)ethan-1-one
(2E)-3-(4-methoxyphenyl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzenesulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(6-cyclopropylpyrimidin-4-yl)pyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
4-cyano-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrrole-2-carboxamide
9-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
3-methyl-8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one