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N-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-methylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-{2-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}acetamide
6-[(2-hydroxy-4-methoxyphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
(2S,4R)-N-(furan-3-ylmethyl)-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-propanoyl-4-(3-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({3-methyl-7-[2-(2-methylphenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,2-oxazole-3-carboxamide
2-(piperidine-1-carbonyl)-6-(1H-pyrazol-3-yl)pyrazine
2-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]-2-(4-hydroxyphenyl)acetic acid
1-[(4-chlorophenyl)methyl]-N-[(3-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-carboxamide
(1S,2S,9R)-11-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(3-phenylpropyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxolan-3-yl)acetamide
2-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethoxy)ethan-1-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
methyl (1R,3S,3aR,6aS)-5-methyl-3-[3-methyl-4-(pyrrolidin-1-yl)phenyl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3S,7S,8aS)-3-(4-aminobutyl)-7-[(thiophen-3-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(2-{[3-(5-methylfuran-2-yl)phenyl]formamido}ethyl)piperidine-3-carboxamide
1-{6-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
N-{2-[(2-ethylphenyl)carbamoyl]ethyl}-3-(1,2-oxazinan-2-yl)propanamide
2-[1-(2,2-dimethylpropyl)-4-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
5-[(3-hydroxy-2,2-dimethylpropyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-amino-6-[2-(propan-2-yloxy)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
8-[(4-methoxypyridin-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-methylbut-2-en-1-yl)-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(piperidine-1-carbonyl)-N-(propan-2-yl)pyrazine-2-carboxamide
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
5-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
3-methyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
3-cyclopentyl-N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}propanamide
1-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
4-[2-(morpholin-4-yl)benzoyl]piperazine-2-carboxylic acid
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
(3R,5S)-N-(4-fluorophenyl)-1-(2-phenylethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(4-fluorophenyl)ethyl]piperidine-3-carboxamide
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidine-3-carboxylate
1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]urea
dimethyl(3-{2-[1-(2-methylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
5-[4-(3-methoxypropyl)piperidine-1-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2,1,3-benzoxadiazole
(1R,2R,6S,7S)-4-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-(1H-indol-3-yl)-1-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl}propan-1-one
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-acetyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)piperidine-3-carboxamide
ethyl 2-{1-[2-(2-phenylethyl)-1,3-benzoxazole-5-carbonyl]piperidin-2-yl}acetate