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6-[4-(ethanesulfonyl)piperazin-1-yl]-N2,N2-diethylpyrimidine-2,4-diamine
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-{2-[3-(2H-1,3-benzodioxol-5-yl)phenoxy]ethyl}-1H-imidazole
N-benzyl-N-[(3-methylpyridin-2-yl)methyl]morpholine-2-carboxamide
6-[cyclohexyl(methyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-methyl-4-(4-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}phenyl)butan-2-ol
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethyl-N,2,3-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-(5-aminopyridin-3-yl)-N-tert-butylfuran-2-carboxamide
2-phenyl-N-({7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-(3,5-dimethylphenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-2-one
2-phenyl-1-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1H-imidazole
N-(2-fluoro-5-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})carbamoyl]amino}phenyl)acetamide
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
5-benzyl-5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide
(2S,4S)-N-ethyl-1-[(4-fluoro-2-methylphenyl)methyl]-4-(3-methoxypropanamido)pyrrolidine-2-carboxamide
methyl 3-cyclopentanecarbonyl-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl (2S)-1-[(4-{[4-(propan-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]pyrrolidine-2-carboxylate
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(furan-2-yl)benzamide
methyl 3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[(cyclopent-3-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
(2S)-1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-3-phenylpropan-1-one
[(4S)-4-amino-5-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-5-oxopentyl]urea
N-[1-(4-{[(2-benzyl-1,3-thiazol-4-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
methyl[(2-methyl-1H-imidazol-4-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
1-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[5-(2,3-dichlorophenyl)furan-2-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
N-({1-[(4-fluorophenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-(4-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)prop-2-yn-1-ol
N-cyclopropyl-3,5-dimethyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1,2-oxazole-4-sulfonamide
1-(4-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
3-[(3-methoxyphenyl)methyl]-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-(1H-indol-3-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]butanamide
N-[4-(2-fluorophenoxy)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-2-carboxamide
3-tert-butyl-1-({1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl}methyl)urea
9-(2-methyl-6-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N-(cyclobutylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{4-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)thiomorpholine
[9-(3-ethyl-1H-pyrazole-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(2-phenoxyethyl)acetamide
N,N-dimethyl-5-[2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-cyclopentyl-1-(2-methylpropyl)-5-[3-(2-oxopyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-phenylpropyl)propanamide
4-methyl-6-(4-{[2-(2-methylphenyl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[2-(pyrrolidine-1-sulfonyl)ethyl]amine
1-[(cyclopropylcarbamoyl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid