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2-(5,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
N-(1,3-dihydroxypropan-2-yl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
7-fluoro-3-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
5-methoxy-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-4-oxo-4H-pyran-2-carboxamide
1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(1R,5S,6S)-6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
N-(2-methoxyethyl)-4-methyl-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}benzamide
N-[(2R,3R)-1'-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}azetidin-3-ol
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-methanesulfonylpiperazine
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carbonitrile
ethyl 1-[3-({[(3-chlorophenyl)methyl]amino}methyl)-8-methylquinolin-2-yl]piperidine-4-carboxylate
1-(2-methoxyethyl)-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
N-[1-ethyl-5-(4-ethylpiperazine-1-carbonyl)-2-(2-fluorophenyl)-1H-1,3-benzodiazol-7-yl]acetamide
5-butyl-1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methoxyphenyl)ethan-1-one
5-(pyridin-3-yl)-5-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)imidazolidine-2,4-dione
N-methyl-1-(4-methylquinazolin-2-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
N-(4-fluorophenyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-amine
(1R,2R,4R)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoacetamide
[(2S,6S)-11-methoxy-4-[3-(methylsulfanyl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-(3-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-1,2,4-triazole
5-(1-benzoxepin-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
9-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
2-[3-(1,3-benzothiazol-2-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]benzamide
4-(5-cyclopropyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperazine-1-carbaldehyde
4-[3-(methylsulfanyl)propanoyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
(3aR,6aR)-2-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-3-amine
4-{[2-(4-hydroxyphenyl)-1H-imidazol-1-yl]methyl}-N,N-dimethylbenzene-1-sulfonamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-amine
1-(4-fluorophenyl)-6,6-dimethyl-N-(1-propylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-hydroxy-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(phenylamino)pyrimidine-5-carboxamide
(4aS,8aR)-6-(5-ethyl-1,3-oxazole-4-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-chloro-4-fluoro-N-methyl-N-(pyrazin-2-ylmethyl)-1-benzothiophene-2-carboxamide
3-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-N-[(3-methyl-7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
4-{2'-amino-3'-cyano-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-4'-yl}benzamide
N-[3-(3-hydroxypiperidin-1-yl)propyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide