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(3R,4S)-N,N-dimethyl-4-(propan-2-yl)-1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-amine
1-benzyl-6-methoxy-4-(5-phenyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-2-one
1-cyclohexyl-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(3,4-dichlorophenyl)morpholine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-propoxyacetamide
4-{1-[6-(4-methylphenyl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
methyl 3-(2-ethylbutyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-{4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-8-methylquinolin-2-yl}-1H-pyrazol-1-yl)ethan-1-ol
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)thian-4-amine
1-oxo-N-(oxolan-3-ylmethyl)-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
2-(3-methoxypropyl)-9-[(5-propylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinolin-4-ol
4-{[3-(5-methoxypyridin-3-yl)phenyl]methyl}morpholine
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
5-{[4-(1-benzofuran-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethylpyrimidine
(1S,5R)-3-(4-methylpiperazine-1-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamide
3-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
4-(benzyloxy)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]cyclopropanecarboxamide
N-{2-[methyl(phenyl)amino]propyl}thian-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(cyclopropylmethyl)amino]piperidin-1-yl}benzamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
4-{[3-(dimethylamino)propyl]amino}-5-methyl-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-4-methyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
5-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-oxo-4-[4-(2-phenylethyl)piperidin-1-yl]butane-1-sulfonamide
3-(3-chlorophenyl)-3-[(2-ethylpyrimidin-5-yl)formamido]propanoic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
ethyl 1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
N,N-dimethyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazin-2-amine
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]pyrrolidin-2-one
2-{5-[3-(trifluoromethyl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
6-[4-(2-fluorophenyl)benzoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(3-methylbutyl)-2-oxo-3-(pyridin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
(3S,4R)-1-[(2,3-dichlorophenyl)methyl]-3-methoxypiperidin-4-amine
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
N-({7-[3-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(piperidin-1-yl)ethan-1-one
1-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(4-aminopyrimidin-2-yl)-4-(1H-indol-2-ylmethyl)-1,4-diazepan-6-ol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methoxybenzamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
(3S,4S)-4-(morpholin-4-yl)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-ol
N-[2-(dimethylamino)ethyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4S)-4-cyclopropyl-1-[2-(4-fluorophenyl)benzoyl]pyrrolidin-3-amine
2,4-difluoro-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide