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3-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl]propanoic acid
4-[(4-hydroxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(5-fluoropyrimidin-2-yl)-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
1-methyl-N-[(4-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}pyridine-3-carboxamide
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2,3,6-trifluorobenzamide
2,6-dimethyl-4-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
2-(2H-1,3-benzodioxol-5-yl)-N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}acetamide
N-{[7-(2,4-dimethylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
N-[(2R,3R)-1'-[(3-fluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
1-[5-(cyclohex-3-en-1-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
4-(4-methyl-2-oxo-2H-chromen-7-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2,4-dichlorophenoxy)-1-[3-(piperidin-1-yl)azetidin-1-yl]ethan-1-one
N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
1-(4-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}thiophen-2-yl)ethan-1-one
3-{1-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-imidazol-2-yl}pyridine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1H-pyrazole-4-sulfonyl)piperidin-3-yl]propanoic acid
3,5-dimethyl-4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
(3aS,6aS)-2-cyclopentanecarbonyl-5-[6-(methoxymethyl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(4-fluoro-2-methylphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
5-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-{6-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]pyrimidin-4-yl}piperidin-4-ol
N-{4-[1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
N-(adamantan-1-ylmethyl)-N-methyl-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
2-ethyl-9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidin-4-ol
1-[1-(3-phenylpiperidin-1-yl)propan-2-yl]-1H-1,3-benzodiazole
N-[(3,4-dichlorophenyl)methyl]-N-methyloxan-4-amine
1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-methanesulfonylacetamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
1-(6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-yl)azepane
N-[(1-methylpiperidin-4-yl)methyl]-2-(1H-pyrazol-1-yl)acetamide
N-methyl-N-(pentan-3-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,2-dimethylpropyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-ethyl-5-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1,2-oxazole
2-[3-(2-methoxyethyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
1-(4-{2-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
(2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-4-yl)methanol
2-methoxy-2-phenyl-N-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methyl-1-(2-phenylethyl)piperidin-3-amine
(2E)-3-(3-fluorophenyl)-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]prop-2-enamide
2-oxo-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,2-dihydroquinoline-4-carboxamide