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1-(4-amino-5-cyanopyrimidin-2-yl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-(dimethylamino)-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}benzamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
N-[3-(furan-2-yl)propyl]-2-methyl-1,3-benzothiazole-6-carboxamide
5-[2-(cyclopropylcarbamoyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
(2S,4R)-1-benzyl-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-amine
1-methyl-6-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}pent-4-enamide
5-({2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
1-(3,5-dimethylphenyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-2-one
(5S,9aS,9bS)-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-4-(morpholin-4-yl)butan-1-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(dimethylamino)-N,4-dimethylpyrimidine-5-carboxamide
N,N,4-trimethyl-6-[4-({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]pyrimidin-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-(2,3,4-trifluorobenzoyl)-1,4-diazepane
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1-propylcyclopropyl)amino]methyl}piperidin-2-one
dimethyl(2-{2-[1-(pyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
6-methyl-5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]quinoline
1-(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-2-phenylethan-1-ol
N-(4-chloro-3-methoxyphenyl)-2-{[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]amino}acetamide
2-amino-N-methyl-6-(2-methylpropyl)-N-[(3-methylpyridin-2-yl)methyl]pyrimidine-4-carboxamide
2-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}pyrazine
5-[3-(2-ethoxyethyl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
6-(morpholin-4-yl)-N-[3-(pyridin-4-yl)propyl]pyrimidin-4-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
1-{4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
(3S,4R)-1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(5-chloro-3-methoxy-2-propoxyphenyl)methyl]-1,4-diazepane
8-[(2-ethylpyrimidin-5-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-methyl-4-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}butan-2-ol
3-({[(2-fluorophenyl)methyl][2-(4-methoxyphenyl)ethyl]amino}methyl)piperidin-3-ol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-methyl-3-phenyl-1H-pyrazole-5-carboxamide
4-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}thiomorpholine
(3aS,6aS)-2-cyclopentyl-5-(3,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
4-(2H-1,3-benzodioxol-5-yl)-2-methylquinoline
1-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)urea
2-oxo-6-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
7-(2-fluoro-4-methylbenzoyl)-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
N-(1-hydroxybutan-2-yl)-2-(phenylformamido)-N-(thiophen-2-ylmethyl)acetamide
(3R)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3,4,4-trimethylpyrrolidin-3-ol
2-{4-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonane-7-carbonyl]piperidin-1-yl}acetamide
ethyl 4-[({6,7-dimethoxy-1-[(4-methylphenyl)methyl]-2-oxo-1,2-dihydroquinolin-3-yl}methyl)amino]piperidine-1-carboxylate
3-(propan-2-yl)-1-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)urea
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(quinolin-8-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate