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1-cyclopentanecarbonyl-N-(isoquinolin-5-ylmethyl)-N-methylpiperidine-4-carboxamide
N,N,7-trimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
1-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)piperidin-4-ol
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
8-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,2,3,4-tetrahydroquinoline
2-methanesulfonyl-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
(2R,6R)-4-[2-(ethanesulfonyl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(5S,9aS,9bS)-5-(1-ethyl-1H-1,3-benzodiazol-2-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{9-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-{[4-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(oxolan-2-ylmethyl)quinoline-2-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(4-methoxyphenoxy)piperidine
3-({[1-(4-fluorophenyl)piperidin-4-yl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
4-(2-ethoxyphenyl)-7-methylthieno[3,2-d]pyrimidine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(2-hydroxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
3-chloro-2-methyl-N-[3-(pyridin-3-yloxy)propyl]benzamide
6-fluoro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[5-(6-oxo-1,6-dihydropyridin-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
3-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}-1-methyl-1,2-dihydroquinolin-2-one
2-(2-methoxy-5-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(2-methylphenyl)propanamide
[1-(2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-3-methyl-1H-pyrazol-1-yl}ethyl)piperidin-4-yl]methanol
6-methoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1H-indazol-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
1-(furan-3-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-methylurea
5-methyl-1-(4-methylphenyl)-4-(quinoxaline-6-carbonyl)piperazin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxy-2-phenylacetamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4,5-dimethyl-2-(2-methylpropanamido)thiophene-3-carboxamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,5-dimethylpyrimidine
2-(2-methoxy-4-methylphenoxymethyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
6-(2-methylpropyl)-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyrimidin-2-one
2-[5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyrazine
3-(2,4-dimethoxyphenyl)-6-methylpyridin-2-amine
1-ethyl-4-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(furan-3-carbonyl)piperidine-4-carboxylic acid
(5S,9aS,9bS)-5-(3-chlorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2-{4-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)pyridine
8-chloro-2-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]quinoline
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-4-(morpholin-4-yl)pentan-1-one
(1R,3S)-3-{[(4-methoxyphenyl)methyl](pyridin-2-ylmethyl)carbamoyl}cyclopentane-1-carboxylic acid
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-[(3-methoxyphenyl)amino]-N-methylbutanamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-{3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione