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N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-1,3-thiazole-5-carboxamide
N-{5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]pyridin-2-yl}methanesulfonamide
3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyridine
methyl({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})(pyrazin-2-ylmethyl)amine
4-(3-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(piperidin-4-yl)pyridine-3-carbonitrile
5-(morpholin-4-ylmethyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}furan-3-carboxamide
1-(2,4-difluorophenyl)-5-(1-propoxyethyl)-1H-1,2,4-triazole
3-[5-(4-methylpentyl)-1,2,4-oxadiazol-3-yl]pyridazine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
(3R,5R)-N-[2-(dimethylamino)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]piperidine-3-carboxamide
3-ethyl-1-methyl-N-[2-(phenylsulfanyl)ethyl]-N-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(3,3-difluoropiperidin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-(piperidin-3-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
(2E)-3-(pyridin-2-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}prop-2-enamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(pyrazin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
3-(1-methyl-1H-pyrrol-2-yl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
(1S,6R)-N-(3-chlorophenyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
[(2-chloro-3,4-dimethoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-(pyrrolidin-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
(3S)-2-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylic acid
1-[(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenylpiperidine
methyl 4-[4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazin-1-yl]benzoate
2-(2,2-diphenylethyl)-4-(oxane-4-carbonyl)morpholine
2-(3-chloro-4-hydroxyphenyl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3-(4-benzoylpiperazine-1-carbonyl)-6-phenyl-1,2-dihydropyridin-2-one
1-(3-ethyl-1,2-oxazole-5-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
1-[(3-methyl-1H-indol-2-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
4-[2-(3-{[(2R)-2-methylpiperazin-1-yl]methyl}phenoxy)ethyl]morpholine
3-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[(3R,4S)-1-(2-carbamoylethyl)-4-propylpyrrolidin-3-yl]-5-chlorothiophene-2-carboxamide
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-ethylpyridine-3-carboxamide
(3S,4S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
2-butyl-5-[4-(pyridin-4-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-benzoxazole
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]propanamide
5-chloro-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1H-indole-2-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
4-[2-(methylsulfanyl)benzoyl]-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3R)-N1-[6-(2-methoxyphenyl)pyridazin-3-yl]cyclopentane-1,3-diamine
N-(2,4-dimethylphenyl)-2-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)acetamide
5-methyl-N4-[(1R,2S)-2-phenylcyclopropyl]pyrimidine-2,4-diamine
N3-butyl-N5-cyclooctyl-N3-methyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-4-{5-[1-(furan-2-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,6-tetrahydropyridine
[(3R,5R)-1-(3-fluoro-4-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
(3aS,6aS)-2-(2-hydroxyethyl)-5-(quinolin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]furan-3-carboxamide
4-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}piperazin-2-one