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N-benzyl-3-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]benzamide
N-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}methanesulfonamide
(3S,4S)-1-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}piperidine-3,4-diol
6-(4-acetyl-1,4-diazepan-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(4-acetamido-3-methoxyphenyl)-5-methyl-1H-pyrazole-3-carboxylic acid
1-(3-carbamoyl-6-methylpyridin-2-yl)-4-phenoxypiperidine-4-carboxylic acid
(4aS,8aR)-1-(3-methoxypropyl)-6-(2-methyl-1-benzofuran-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(dimethyl-1,2-oxazol-4-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)propanamide
3-benzyl-1-methyl-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(3-fluoropyridin-4-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-[(1-methylpiperidin-4-yl)methyl]pyridine-3-carboxamide
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
2-({[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,8aR)-6-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-(azocan-1-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
N-(3,4-dimethylphenyl)-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]acetamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-butyl-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
1-[(8-fluoroquinolin-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2,4-dimethyl-6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}pyrimidine
6-[methyl(pyridin-2-ylmethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
3-methoxy-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyridine-2-carboxamide
3-(2-fluorophenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]-3-phenylpropan-1-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(oxan-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(methylsulfanyl)ethyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
(3R,4S)-1-(5-chloro-2-fluorobenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-amine
9-(2,3,4-trifluorobenzoyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-[(1S)-1-(4-fluorophenyl)ethyl]-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(5-acetylthiophen-3-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-(2-methoxyethyl)-1-(1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
9-(2,6-difluoro-3-methylbenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-(3-hydroxy-3-methylbutyl)-N-[2-methyl-1-(4-methylpiperazin-1-yl)propan-2-yl]benzamide
8-(3-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]thiophene-2-sulfonamide
1-(2,2-diethylcyclopropanecarbonyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-butyl-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(2-{[9-(2-chlorophenyl)-15-methyl-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-12-yl]formamido}ethyl)acetamide
(furan-2-ylmethyl)({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
(1S,4S)-2-(2-chlorophenyl)-5-[(1-methyl-1H-pyrrol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(2-methoxyethoxy)-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethan-1-one
2-(1H-imidazol-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
3-(1-{2-[4-(dimethylamino)phenyl]acetyl}piperidin-3-yl)-N,N-dimethylpropanamide