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2-[3-benzyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide
3-cyclopropyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
(1S,5R)-3-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,6aR)-5-(3-hydroxypyridine-2-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methoxy-5-oxo-6-(3-propoxypropyl)-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-(carbamoylmethyl)-N-[(2,6-dimethylpyridin-4-yl)methyl]piperidine-4-carboxamide
1-(4-chloro-2-ethylphenyl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
4-(benzyloxy)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
2-[cyclopropyl(pyridin-4-ylmethyl)amino]-N-(2-acetamidophenyl)acetamide
2-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
2-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}thiophene-3-sulfonamide
(5S,9aS,9bS)-5-(2,5-dimethoxyphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(butan-2-yl)-2-methyl-N-(pyridin-4-ylmethyl)-5-sulfamoylbenzamide
1-(1-benzofuran-2-ylmethyl)-3-(methanesulfonylmethyl)piperidine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
6-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyridine-3-carboxamide
1-cyclopentyl-3-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)urea
1-(furan-2-yl)-2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethane-1,2-dione
2-(1-methyl-1H-pyrazol-3-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,4-dimethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
8-[3-(methylsulfanyl)propanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
methyl({[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
3-{[7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
9-(2-chloro-5-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-5-{[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]methyl}furan-2-carboxamide
N-methyl-N-(oxan-4-yl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propoxy}benzamide
N4-methyl-N4-(3-phenylpropyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(2,3-dihydro-1H-inden-2-yl)-1-(5-methanesulfonyl-2-methylphenyl)-3-methylurea
N-[3-(2-methylpyrimidin-4-yl)phenyl]-2-(morpholin-3-yl)acetamide
9-(2H-1,3-benzodioxol-5-yl)-15-methyl-N-(3-methylbutyl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
(2S,4R)-4-(cyclooctylamino)-N-methyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N5-cyclopropyl-N6-[(2-phenyl-1,3-thiazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[({4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)methyl]-1λ6-thiane-1,1-dione
1-{3-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
(1S,5R)-3-[4-(1H-imidazol-1-yl)butanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(3,5-difluorophenyl)ethyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2,4-difluorophenyl)carbamoyl]piperidine-4-carboxylate
3-ethyl-5-{3-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-1,2,4-oxadiazole
1-cyclohexyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-4-carboxamide
2-[(5-ethylfuran-2-yl)methyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-tert-butyl-2-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]benzene-1-sulfonamide
2-(3-fluorophenoxymethyl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-1,3-oxazole-4-carboxamide
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
3-(4-phenylbenzoyl)-N-propylpiperidine-1-carboxamide
N-cyclopropyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(thiophen-3-ylmethyl)acetamide