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1-ethyl-2-oxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-dihydropyridine-4-carboxamide
6-methyl-2-{[(3R,4S)-1-(oxane-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
N4-[(1S)-1-phenylethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]ethan-1-one
N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(2R,6R)-4-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-methoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aS,8aR)-6-(2-ethoxypyridine-3-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-ethyl-3-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}urea
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amino)methyl]pyrrolidin-2-yl]methanol
2-(6-methoxynaphthalen-2-yl)-4-(6-phenylpyridazin-3-yl)morpholine
N-[3-(pyridin-3-yl)propyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
2-{[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl](methyl)amino}ethan-1-ol
3-(1-{3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)sulfanyl]propanoyl}piperidin-3-yl)propanamide
5-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-cyclobutanecarbonyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
1-methyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
N-(furan-2-ylmethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
4-(4-{1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenyl)but-3-yn-1-ol
N-cyclohexyl-3-{[(5-methoxy-2-methylphenyl)carbamoyl]amino}propanamide
4-(2-methyl-1H-imidazol-1-yl)-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
5-ethyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4,6-dimethyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(3,5-dimethylphenyl)-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperazin-2-one
(3S,4S)-4-(4-fluorophenyl)-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]piperidin-3-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
N-ethyl-3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carboxamide
N-(butan-2-yl)-N-(pyridin-4-ylmethyl)butanamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,6-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N4-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-5-methylpyrimidine-2,4-diamine
(3S,4R)-1-(4-chloro-2-methylbenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
4-(2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-2-yl}ethyl)morpholine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
5-chloro-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[1-(4-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-yl]methanol
methyl (1S,3S,3aR,6aS)-3-(1-ethyl-1H-imidazol-2-yl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-4-(thiophen-2-yl)butanamide
[(1-benzyl-1H-pyrazol-4-yl)methyl]({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amine
N-cyclopropyl-N-{[2-(2,3-dimethoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamide
2-cyclopentyl-9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-{[methyl(thian-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-propylpyrrolidin-2-one
[(3R,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-cyclohexyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-4-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide