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(2R)-2-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(1H-indol-3-yl)propanamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
7-[(3-ethenylphenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
(3R,4R)-4-ethyl-1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidine-3,4-diol
2-(dimethylamino)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
(1S,5R)-3-(3-chloro-2-fluorobenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-2-{[2-(morpholin-4-ylmethyl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]acetamide
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
2-[4-(trifluoromethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrimidin-2-amine
methyl 4-(5-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
9-[2-(morpholin-3-yl)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(5-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}furan-2-yl)benzonitrile
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-hydroxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]urea
2-(3-methoxypropyl)-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]piperidine
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
7-[2-(pyridin-2-ylsulfanyl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-[4-(ethylcarbamoyl)phenyl]-4-[2-(2-hydroxyethoxy)ethyl]piperazine-1-carboxamide
4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
5-{1-[3-(methylsulfanyl)propyl]-1H-imidazol-2-yl}-2,1,3-benzothiadiazole
N-(3-chloro-4-fluorophenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
1-(1H-imidazol-2-ylmethyl)-3-[2-(3-methoxyphenyl)ethyl]piperidine
9-(3-hydroxypyridine-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(1-butyl-1H-imidazol-2-yl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
ethyl 3-{[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}propanoate
[1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-propylpiperidin-3-yl]methanol
3-(4-hydroxyphenyl)-N-[3-(1H-imidazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
N-[(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
1-cyclopentyl-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
6-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-2-methyl-6H,7H-[1,3]oxazolo[5,4-d]pyrimidin-7-one
1-{1-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)benzamide
(2S,4S)-4-amino-N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-1-methylpyrrolidine-2-carboxamide
N-[(3R)-piperidin-3-yl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
4-{1-cyclohexyl-5-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
N-(1-benzylcyclopropyl)-N'-(2-ethoxyphenyl)propanediamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-[2-(pyridin-2-yl)ethyl]piperazine
1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-(pyridin-2-ylmethyl)urea
1-(4-fluorophenyl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}cyclopropane-1-carboxamide
1,5-dimethyl-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
7-(1-benzothiophen-3-yl)-4-(1-ethylpiperidin-4-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(carbamoylmethyl)-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(2-methoxyphenyl)-N-[3-(pyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide