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(1S,5R)-3-benzyl-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-methanesulfonyl-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl 3-{[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}propanoate
N-benzyl-2-[4-(4-{[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
4-ethyl-3-{1-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
4-(1,2,3,4-tetrahydronaphthalen-2-yl)-N-(1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
1-[(3,5-difluorophenyl)methyl]-4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazine
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2,6-dimethylquinoline-4-carboxamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(1-methylpiperidin-4-yl)acetamide
(1R,5R)-6-methyl-3-(2,4,5-trifluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
6-{[(2S,5R)-5-(1,4-oxazepan-4-ylmethyl)oxolan-2-yl]methyl}quinoline
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
3-(2-methoxyphenyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
(2-{2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-benzyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(2-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenoxy)ethan-1-ol
1-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one
N-methyl-N-{[2-(methylsulfanyl)phenyl]methyl}oxan-4-amine
5-(2,6-difluorophenoxymethyl)-N-[(3,4-dimethoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
1-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-butyl-4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-methylpiperazin-2-one
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-4-acetamidobutanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(3aR,7aS)-2-{4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
6-methyl-2-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
N-[(1R,2R)-2-hydroxycyclohexyl]-6-methoxy-3-methyl-N-propyl-1-benzofuran-2-carboxamide
ethyl 4-[3-(cyclopropylcarbamoyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine-1-carboxylate
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-{[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,3-oxazolidin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
4-[4-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]but-3-yn-1-ol
2-amino-1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-ethyl-7,8-dimethyl-N-(propan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
1-phenyl-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pentane-1,5-dione
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(furan-2-yl)-4-phenylbutan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
5-methoxy-2-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]pyridin-4-ol
4-{1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-methoxypropyl)-9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-oxoethyl}-1H-indole-3-carboxamide