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8-[2-(pyrrolidin-1-yl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)pyridine
N-butyl-4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
1-acetyl-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-3-[2-(methoxymethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
{3-[(3-chlorophenyl)methyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methanol
1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
6-(2-chlorophenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
{3-[2-(2-chloro-3,4-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}methanol
2-[5-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-phenylethane-1,2-dione
{3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]phenyl}methanol
(4aS,8aR)-1-(2-methylpropyl)-6-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-decahydro-1,6-naphthyridin-2-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(propane-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
5-methoxy-1,2-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-indole-3-carboxamide
4-(4-chloro-3-methylbenzoyl)-1-(2-methoxyphenyl)-5-methylpiperazin-2-one
5-(3-fluorophenoxymethyl)-N-(1-hydroxybutan-2-yl)-1H-pyrazole-3-carboxamide
3-{[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]methyl}benzoic acid
2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-3-carboxamide
1-[(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-4-methylpiperazine
(2E)-3-(4-methoxyphenyl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]prop-2-enamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-phenyl-1,2-oxazole-3-carboxamide
2-(3-chlorophenoxy)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(6-methylpyridine-2-carbonyl)piperidine-4-carboxamide
1-(azocan-1-yl)-3-[5-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-[(5-ethylpyridin-2-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
(3aR,5S,6S,7aS)-2-[(3-methylthiophen-2-yl)sulfonyl]-octahydro-1H-isoindole-5,6-diol
4-(2-methylpyrimidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S,4S)-4-[3-(benzenesulfonyl)propanamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(1H-1,2,3,4-tetrazol-5-ylmethyl)amino]pyridine-3-carboxamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
3-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-9-methyl-3,9-diazaspiro[5.6]dodecane
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-thiazole-4-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
1-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]pyrrolidin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(4-chlorophenyl)-5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-1,2,4-oxadiazole
N-(6-chloro-2-methylpyridin-3-yl)-4-[(3,5-difluorophenyl)methyl]piperazine-1-carboxamide
3-{[4-(3-chlorophenyl)-5-{[methyl(thiophen-2-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{1'-[2-(morpholin-2-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
5-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-methyl-4-{1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrazolo[1,5-a]pyridine-3-carboxamide
1-methyl-3-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-{3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenoxy}acetamide
(2S)-2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylformamido]-3-(4-hydroxyphenyl)propanamide
N4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylsulfanyl)pyrimidine-4,6-diamine