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3-[(2R,3R,6R)-5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(azepan-1-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
3-(3,4-dimethylphenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
methyl 3-(4-{[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
4-[(2S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carbonyl]morpholine
2-(3-{3-[5-(piperidine-1-carbonyl)furan-2-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
1-(3-methylfuran-2-carbonyl)spiro[azepane-4,2'-chromene]
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-(cyclohexylmethyl)-N5-(1,2-diphenylethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
3-methyl-1-[3-(4-methylpiperidine-1-carbonyl)phenyl]-3-(oxolan-3-ylmethyl)urea
2-(benzylsulfanyl)-N4-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-4,6-diamine
N4-methyl-N4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-3-carboxylate
(3aS,6aR)-5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-methyl-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{3-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
4-{4-[(1H-imidazol-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
2-(4-methylphenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
1-(furan-2-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,3R)-N1-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
(1R,3s,6r,8S)-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(5-methyl-1,3-thiazol-2-yl)benzamide
9-(2-hydroxyethyl)-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-[(4-methyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
5-{4-phenyl-1-[1-(thiophen-2-yl)propyl]-1H-imidazol-5-yl}pyrimidin-2-amine
(3S)-3-ethyl-4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]morpholine
2-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
2-(cyclohexylmethyl)-4-(2-methoxypyridine-3-carbonyl)morpholine
4-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-5-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)naphthalene-1-carboxamide
3-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
3-(1-ethyl-1H-imidazol-2-yl)-1-[2-(2-ethylphenoxy)ethyl]piperidine
8-(2-methoxypyridine-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-3-phenyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-4-carboxamide
4-[({6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1-ethylpyrrolidin-2-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine
[(4-fluorophenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine