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N-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
2-[({5-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
4-[(3-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]morpholine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
3-(3-fluorophenyl)-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1,2,4-oxadiazole
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(thiophen-2-ylmethyl)propanamide
3-(3,4-difluorophenyl)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-2,5-dihydro-1H-pyrrole
N-[(3R,4S)-4-cyclopropyl-1-(4-methoxypyrimidin-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
1-(4-{1-[1-(3-methylpyridin-2-yl)propyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)ethan-1-one
(2S)-1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(dimethylamino)-4-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidine-5-carboxamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
2-(4-chlorophenyl)-4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}morpholine
butyl 3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-cyclopropyl-5-(6-oxo-1-propylpiperidine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(3-cyano-4-methylphenyl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(furan-2-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
4-(2-ethoxyethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)imidazolidine-2,4-dione
3-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
(3S,4S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
8-methyl-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(3S)-2-oxoazepan-3-yl]benzamide
4-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
ethyl 4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
N-ethyl-6,8-dimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
methyl 2-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}amino)acetate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-(propan-2-yl)-2-({6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazol-3-yl}formamido)acetamide
4-[5-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
(5-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}furan-2-yl)methanol
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
methyl (2S,4S)-4-(5-chlorothiophene-2-sulfonamido)-1-methylpyrrolidine-2-carboxylate
N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-5-ethyl-1,3-oxazole-4-carboxamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2-methoxyphenyl)ethan-1-one
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
N-{4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}acetamide
N-{2-[(pyridin-3-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5R)-6-(2-chloro-4-fluorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(3-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-{[(4-phenyloxan-4-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
(2S)-1-[3-(cyclobutylcarbamoyl)benzenesulfonyl]-N-ethylpyrrolidine-2-carboxamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide