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2-[1-(2,2-dimethylpropyl)-4-[1-(furan-2-ylmethyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)piperidin-2-one
4-[5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carbonyl]morpholine-2-carboxamide
3-(methoxymethyl)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(oxan-2-yl)ethyl]acetamide
5-[1-(cyclohex-3-en-1-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
2,5-dioxo-6-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
6-(2-chloro-6-fluoro-3-methylphenyl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
methyl 6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-[(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-(2-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-(thiophen-3-ylmethyl)piperidine
2-methoxy-N-methyl-5-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzamide
1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
(1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(1H-indazol-7-yl)urea
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
4-(hydroxymethyl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-ol
4-{3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]phenyl}-4H-1,2,4-triazole
1-[4-(oxolane-2-carbonyl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
N-methyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
3-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-{[methyl({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)amino]methyl}pyridine-3-carboxylic acid
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)pyridine-4-carboxamide
N-butyl-2-(dimethyl-1,2-oxazol-4-yl)-N-(thiophen-3-ylmethyl)acetamide
(3R,4S)-3,4-dimethyl-1-(2-methyl-4-phenylpyridine-3-carbonyl)piperidin-4-ol
6-methoxy-2-oxo-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
6-(2-ethyl-1H-imidazol-1-yl)-2-methylquinolin-4-ol
N-[(4-fluorophenyl)methyl]-3-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}propanamide
({5-[1-(5-chloro-3-fluoropyridin-2-yl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]acetic acid
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-(piperidine-1-carbonyl)phenyl]urea
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
N-(5-methoxy-2-methylphenyl)-4-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
4-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-6-methyl-2-propylpyrimidin-4-amine
4-methyl-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}azepan-4-ol
2-({2-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
4-{2-[1-(pyridin-4-ylmethyl)piperidin-2-yl]ethyl}phenol
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
ethyl 4-(1-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-cyclopentanecarbonyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)piperidine-4-carboxamide