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4-[3-(1H-indol-3-yl)propanoyl]piperazine-2-carboxylic acid
4-[3-(3,4-dimethylphenyl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
(3R,4R)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
[2-(2-ethoxyphenoxy)ethyl](methyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
4-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
5-(azepan-1-yl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2,6-dimethyl-8-{[1-(thiophen-3-yl)propan-2-yl]amino}octan-2-ol
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(3-methylquinoxalin-2-yl)methyl]amine
N-[(1R,3R)-3-aminocyclopentyl]-2-methyl-4-phenylpyridine-3-carboxamide
(1R,3S,5S)-8-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}-8-azabicyclo[3.2.1]octan-3-ol
4-ethyl-3-{1-[(8-methylquinolin-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(2E)-3-phenylprop-2-enoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-4-({5-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
4-{1-[1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
3-cyclohexyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
1-(4-fluorophenyl)-4-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
N-cyclopropyl-2-methyl-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[2-(thiophen-3-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(1S,5R)-3-benzyl-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole
2-(2H-1,3-benzodioxol-5-yl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}furan-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-[2-({[2-(2-amino-1,3-thiazol-4-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
3-(4-fluorophenoxymethyl)-1-(4-methyl-1,3-thiazol-2-yl)piperidine
(1H-1,3-benzodiazol-2-ylmethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
2-amino-N-[2-(1-benzothiophen-3-yl)phenyl]acetamide
N-[(3-methylphenyl)methyl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(propan-2-yl)acetamide
6-(1-methyl-1H-imidazol-2-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyridazin-3-amine
{1-methyl-4-[6-(propan-2-yl)pyrimidin-4-yl]piperazin-2-yl}methanol
N-(3-hydroxypropyl)-2-methyl-N-(pyridin-3-ylmethyl)-1-benzofuran-7-carboxamide
N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-methyl-4-(pyrrolidine-1-carbonyl)-N-(quinolin-5-ylmethyl)pyridin-2-amine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-ethyl-5-(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)imidazolidine-2,4-dione
N3-cyclooctyl-1-(2-methoxyethyl)-N5-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(but-2-ynoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,2-oxazole-3-carboxamide
4-(3-fluorophenoxy)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
2-chloro-N-[(3-methylthiophen-2-yl)methyl]-5-(1H-pyrazol-1-yl)benzamide
2-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
dimethyl(3-{2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N-(3,4-difluorophenyl)-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-3-amine
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-5-propyl-1,2-oxazole-3-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one