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3-cyano-N-[6-(3-methoxyphenoxy)pyridin-3-yl]piperidine-1-carboxamide
2-(2-{1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
4-(1,4-diazepan-1-yl)-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-[(3-fluorophenyl)methyl]-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
6-fluoro-2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-2-one
2-butyl-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
1-cyclopropyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
4-(2,4-diethoxy-3-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-oxa-7-azaspiro[4.5]decane
4-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-{1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}benzoic acid
2-(4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-methyl-6-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{3,5-dimethyl-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrazol-4-yl}propanoic acid
2-cyclopropanecarbonyl-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(3,5-dichloro-4-methylbenzoyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
4-(6-methoxynaphthalen-2-yl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-(morpholin-4-ylmethyl)-4H-pyran-4-one
1-[3-chloro-2-(propan-2-yloxy)phenyl]-3-methyl-3-[1-(1,2-oxazol-3-yl)ethyl]urea
(1R,4S)-1,7,7-trimethyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
2-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-methyl-1,3,4-thiadiazole
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})(2-phenylethyl)amine
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4,4-difluoropiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
(3-{2-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-(4-methoxy-2-methylphenyl)-3-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole
1-methyl-5-(morpholin-4-yl)-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(2-{[methyl(oxan-2-ylmethyl)amino]methyl}phenoxy)acetic acid
3,5-dimethyl-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
ethyl 4-benzyl-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxylate
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-(piperazin-1-yl)ethan-1-one
N-(2-hydroxyethyl)-5-{5-methylthieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[5-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]-N-(thiophen-3-yl)piperidine-1-carboxamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-(1-methyl-6-oxopiperidin-3-yl)pyrimidine-5-carboxamide
2-methyl-N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-(4-fluorophenyl)-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1,4-diazepane
4-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-chloro-N-(2-methoxyethyl)-4-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide