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1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one
2-{2-[2-(1-phenyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]ethyl}pyridine
N-{5-[2-(benzyloxy)ethyl]pyridin-2-yl}acetamide
3-(dimethylamino)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[(4-acetamidophenyl)methyl]-2-{[1-(1H-1,2,4-triazol-5-yl)ethyl]amino}acetamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(5-methoxy-5-oxopentanoyl)piperidine-3-carboxylate
2-(1H-imidazol-2-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
2-(1H-indazol-1-yl)-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
3-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-(pyridin-3-yl)propanamide
N-butyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-acetyl-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]thiophene-3-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2-methylpropyl)piperidine-3-carboxamide
2-methyl-5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
(3S,4R)-1-(2-acetamidoacetyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[2-(pyridin-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5-methylpyridine-3-carboxamide
2-{4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N-[3-(cyclopentyloxy)propyl]-6-ethylpyrimidin-4-amine
5-{1-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1H-imidazol-2-yl}-2-methoxyphenol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-5-oxopyrrolidine-3-carboxamide
1-(5-cyanopyridin-2-yl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
1'-(4-methoxybenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(propan-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-hydroxy-2-(4-methoxyphenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
3-{4-[4-(3-methoxypiperidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
4-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-propylpyrrolidin-2-one
methyl 3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
3-(2-amino-1,3-thiazol-4-yl)-1-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-ethyl-N-methyl-4-{1-[3-(methylamino)propyl]-4-phenyl-1H-imidazol-5-yl}aniline
4-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]morpholine
1-(2-aminoethyl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-(cyclopropylsulfamoyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
(3R,5S)-N3-[(dimethyl-1,2-oxazol-4-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
7-methoxy-3-[5-(methoxymethyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
N-[2-(2-fluorophenoxy)ethyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
N,N-dimethyl-4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperazine-1-sulfonamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylic acid
3-ethoxy-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridazine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4,6-dimethoxypyrimidin-2-yl)piperidin-3-ol
2-methyl-1-{4-[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]piperidin-1-yl}propan-1-one
N-[2-(3-fluorophenyl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-(4-aminoazepan-1-yl)-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propan-1-one
({3-[(dimethylamino)methyl]phenyl}methyl)(methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-{2-[methyl(phenyl)amino]ethyl}-3-(1-methylpiperidin-3-yl)propanamide
1-ethyl-N-[(2-methoxyphenyl)methyl]-4,6-dimethyl-2-oxo-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide