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N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
ethyl 1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-2-carboxylate
(4aS,7aR)-1-(3-ethoxypropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(5-methoxyfuran-2-carbonyl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-hydroxy-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N,N-dimethyl-3-{[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]sulfamoyl}benzamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(3-fluorophenyl)propanamide
4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-1H-pyrrole-2-carbonitrile
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(morpholin-4-yl)propyl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
3-methyl-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-(propan-2-yl)acetamide
5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-(3-methylphenyl)pyrimidine
1-[4-({[2-(3-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(5-{1-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
4-methyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
2-methoxy-4-{[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}phenol
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-methyl-2-phenylpiperazine
3-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamido]-4-(3-methylpiperidin-1-yl)benzamide
N-{1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1-oxopropan-2-yl}propanamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-[2-(2,2-diethylmorpholin-4-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[5-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
4-(5-methylfuran-2-yl)-1-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
(3S,4S)-4-(4-fluorophenyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-6-phenylpyridine-3-carboxylic acid
N-[(5-ethylpyridin-2-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-propylacetamide
[(3R,4R)-1-[(3,5-dimethylphenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
2-cyclohexyl-5-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidine
N-[(3S,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-(2-hydroxyphenoxy)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)acetamide
{2-[3-(pyridin-3-yl)azetidin-1-yl]-1,3-thiazol-4-yl}methanol
2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2-dihydrophthalazin-1-one
3-benzyl-5-[5-(methoxymethyl)furan-2-yl]-1,2,4-oxadiazole
3-[(1-cyclobutylethyl)amino]-N-(2,3-dihydro-1H-inden-2-yl)-5-[(propan-2-yl)sulfamoyl]benzamide
N-{2-[3-(thiomorpholine-4-carbonyl)benzenesulfonamido]ethyl}acetamide
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-2-[(prop-2-en-1-yl)amino]benzamide
4-[(3-hydroxypiperidin-1-yl)methyl]-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
4-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-{1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(2-methylpropyl)piperidin-4-amine
9-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
11-[2-(prop-2-yn-1-yloxy)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3,5-difluoropyridine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one