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2-(3-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-3-phenyl-1H-1,2,4-triazol-1-yl}-3-methylpyridine
ethyl 2-{1-[(2-aminopyridin-3-yl)methyl]piperidin-2-yl}acetate
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
1-(cyclohexylmethyl)-N-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]acetamide
1-(2,6-dimethylpyridin-4-yl)-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
[4-ethyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]methanol
N-(2-methoxypropyl)-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
3-(azepane-1-carbonyl)-5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole
methyl (3S)-3-amino-4-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanoate
8-cyclohexyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]acetamide
1-(2,3-dimethoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(2S)-1-methoxypropan-2-yl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
2-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
(4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}morpholin-2-yl)methanamine
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-2-(1-methylpiperidin-4-yl)acetamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2-fluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-2-phenylmorpholine
2-(cyclopropylmethyl)-9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-(methylamino)propan-1-one
3-{2-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
4-(4-{[3-(2-hydroxyethoxy)phenyl]methyl}-5-methyl-2-oxopiperazin-1-yl)benzonitrile
N-[2-(1H-pyrazol-1-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyridin-2-amine
(1R,2S,6R,7S)-4-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-azatricyclo[5.2.2.02,6]undecane
5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-methyl-7-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-ethyl-1-(5-fluoropentyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-[(3-methoxypropyl)sulfamoyl]benzamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-6-ol
N-[(4-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-(1H-imidazol-2-ylmethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}-6-methylpyridin-3-ol
3-(1-propyl-1H-1,2,4-triazol-3-yl)-1-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]urea
1-{1-[(1-ethyl-1H-indol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxylic acid
N,N-dimethyl-7-(3-methylfuran-2-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(2,4-dimethylphenyl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(1-benzofuran-2-yl)-2,5-dimethylpyrimidine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide