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N-[3-({[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(methylamino)benzamide
9-[3-(methylsulfanyl)butyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
(4-{[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}oxan-4-yl)methanol
5-acetyl-2,4-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-pyrrole-3-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-5-oxopyrrolidine-3-carboxylic acid
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
(1R,5R)-3-cyclobutanecarbonyl-6-[(2-fluoro-5-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{[(3-methoxypropyl)amino]methyl}-6,8-dimethylquinolin-4-ol
(3S,4S)-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-ol
2-methyl-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
[(2S,6S)-4-[(5-methylfuran-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-methyl-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1H-pyrazole-5-carboxamide
2-chloro-9-methyl-3-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
4-[(2-hydroxy-3-methoxyphenyl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
1-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-3-(1-methyl-1H-pyrazol-4-yl)urea
(3aS,6aR)-3-cyclopentyl-5-[(3,4-dimethylphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(dimethylamino)-1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(4-methylphenyl)ethan-1-one
2-(methylsulfanyl)-N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
3-[5-(1,1-dioxo-1λ6-thiolan-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
2-chloro-5-acetamido-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
7-(1-benzothiophen-3-yl)-4-[5-(methoxymethyl)furan-2-carbonyl]-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,6R)-3-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
4-amino-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]pyridine-2-carboxamide
N-{2-methoxy-4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}butanamide
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-methyl-6-propylpyrimidine
2-{2-methyl-6-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]pyrimidin-4-yl}ethan-1-amine
2-methoxy-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}acetamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-3-carbonitrile
2-(5-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-yl)benzonitrile
6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxamide
2,6-diamino-4-[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-(4-cyclohexylphenyl)-1-methyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
2-[2-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]pyridine
2-({[(3R,4R)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(dimethylamino)-1-[4-(4-methoxybutyl)piperazin-1-yl]-2-(2-methylphenyl)ethan-1-one
6-methyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
ethyl 1-(2H-1,3-benzodioxole-5-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
4-(cyclopropylmethyl)-1-(2,6-diaminopyrimidin-4-yl)piperidine-4-carboxylic acid
[3-(8-methoxy-2-methylquinolin-5-yl)phenyl]methanamine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-{3-methyl-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-oxobutan-2-yl}acetamide
4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1-phenylpiperazin-2-one
1-cyclopentanecarbonyl-N-[1-(4-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethylpropanamide
2-(furan-2-yl)-N-(2-methoxyphenyl)azepane-1-carboxamide