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3-(azocan-1-yl)-N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]propanamide
1-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-3-ethoxypropan-2-ol
(3S,4S)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-{2-[4-(3-methylphenoxy)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-propyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N,2-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4-phenylpyridine-3-carboxamide
1-(5-chloropyridin-2-yl)-4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
4-[(4-fluorophenyl)methyl]-1-(4-methylpyrimidin-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-cyclooctyl-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1λ6-thiomorpholine-1,1-dione
N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
5-fluoro-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-4-(pyrrolidin-1-yl)pyrimidine
(1S,3R)-3-cyclopropanesulfonamido-N-[2-(4-hydroxyphenyl)ethyl]cyclopentane-1-carboxamide
2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
N-(2-methyl-1-{7-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
4-(2-ethylpyrimidine-5-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-1H-indole
3-(4-methoxyphenyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-methyl-1-(naphthalen-2-yl)urea
4-(3-methoxypyrazin-2-yl)-1H-indole
2-[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]-4,5,6,7-tetramethyl-1H-1,3-benzodiazole
N-methyl-5-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-3-carboxamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(4-fluorobenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-2-(thiophen-2-yl)azetidine
2-fluoro-6-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)phenol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)acetamide
2-(1-{[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
N-butyl-N-(furan-2-ylmethyl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
1-[4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperazine
N-[(3R,4S)-1-cyclohexyl-4-cyclopropylpyrrolidin-3-yl]-3-(pyridin-2-yl)propanamide
9-(2-amino-6-methoxypyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2-{2-[(1-acetylpiperidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-cyclopentyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
6-cyclopropyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
3-[5-(1-carbamoylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopentylpropanamide
3-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-hydroxyethan-1-one
2-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
2-oxo-N-[(1-propylpiperidin-4-yl)methyl]-2-(pyrrolidin-1-yl)acetamide
3-(furan-2-yl)-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-3-phenylpropanamide
1-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-3-benzyl-6-(1-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane